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C127224-5mgMomelotinib (CYT387) is an ATP-competitive inhibitor of JAK1/JAK2 with IC50 of 11 nM/18 nM, ~10-fold selectivity versus JAK3.An inhibitor of JAK1 and JAK2.
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C286575-100mgCytosporone B.
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C128050-10mgCZC24832 is the first selective PI3Kγ inhibitor with IC50 of 27 nM, with 10-fold selectivity over PI3Kβ and >:100-fold selectivity over PI3Kα and PI3Kδ.
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C128050-50mgCZC24832 is the first selective PI3Kγ inhibitor with IC50 of 27 nM, with 10-fold selectivity over PI3Kβ and >:100-fold selectivity over PI3Kα and PI3Kδ.
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