Radiolabeled Receptor Modulators

≥95% (SDS-PAGE):Endotoxin level:Function:On ligand binding, forms a receptor complex consisting of two type II and two type I transmembrane serine/threonine kinases. Type II receptors phosphorylate and activate type I receptors which

Application:Capture antibodyCLIA: 10-40μg/mg BeadsELISA: 1μg/mLLF/GICA : 1mg/mLProtein functionCardiac hormone which may function as a paracrine antifibrotic factor in the heart. Also plays a key role in cardiovascular homeostasis through

Application:Capture antibodyCLIA: 10-40μg/mg BeadsELISA: 1μg/mLLF/GICA : 1mg/mLProtein functionCardiac hormone which may function as a paracrine antifibrotic factor in the heart. Also plays a key role in cardiovascular homeostasis through

Application:Capture antibodyCLIA: 10-40μg/mg BeadsELISA: 1μg/mLLF/GICA : 1mg/mLProtein functionCardiac hormone which may function as a paracrine antifibrotic factor in the heart. Also plays a key role in cardiovascular homeostasis through

Application:Capture antibodyCLIA: 10-40μg/mg BeadsELISA: 1μg/mLLF/GICA : 1mg/mLProtein functionCardiac hormone which may function as a paracrine antifibrotic factor in the heart. Also plays a key role in cardiovascular homeostasis through

Biochem/physiol Actions Rinvanil is a Capsaicin analogue that potently activates transient receptor potential vanilloid 1 (TRPV1) channels. Rinvanil induces neuroprotective mild hypothermia in ischemic brain injured mice through TRPV1 activation.

Biochem/physiol Actions Rinvanil is a Capsaicin analogue that potently activates transient receptor potential vanilloid 1 (TRPV1) channels. Rinvanil induces neuroprotective mild hypothermia in ischemic brain injured mice through TRPV1 activation.

General description RN-9893 is a small, orally bioavailable antagonist of TRPV4 (transient receptor potential subfamily V4. It is a tri-substituted benzamide compound.

General description RN-9893 is a small, orally bioavailable antagonist of TRPV4 (transient receptor potential subfamily V4. It is a tri-substituted benzamide compound.

Biochem/physiol Actions RO5256390 is an orally available partial agonist that targets trace amine-associated receptor 1 (TAAR1) with high affinity (Ki in nM = 0.9/mouse, 4.

Biochem/physiol Actions RO5256390 is an orally available partial agonist that targets trace amine-associated receptor 1 (TAAR1) with high affinity (Ki in nM = 0.9/mouse, 4.

Biochem/physiol Actions RQ-00203078 is an orally available potent and selective TRPM8 antagonist that potently reduces cation currents induced by menthol and other TRPM8 agonists. RQ-00203078 inhibits HSC3 and HSC4 oral squamous carcinoma cell