Protease Inhibitors

RR-11a analog is a potent and irreversible inhibitor of Schistosoma mansoni legumain , with an IC 50 of 31 nM. RR-11a analog is an aza-Asn derivative and aza-peptide Michael acceptorIn VivoRR-11a analog has a half-live of 3-10 min. MCE has not

RR-11a analog is a potent and irreversible inhibitor of Schistosoma mansoni legumain , with an IC 50 of 31 nM. RR-11a analog is an aza-Asn derivative and aza-peptide Michael acceptorIn VivoRR-11a analog has a half-live of 3-10 min. MCE has not

InformationSaxagliptin (BMS-477118) Saxagliptin (BMS-477118, Onglyza) is a selective and reversible DPP4 inhibitor with IC50 of 26 nM.In vitroSaxagliptin has an inhibition constant Ki of 1.3 nM for DPP4 inhibition, which is 10-fold more potent than

Amino Acid Sequence Ser-Phe-Leu-Leu-Arg-Asn-NH2 Application Ser-Phe-Leu-Leu-Arg-Asn-amide trifluoroacetate salt has been used as a protease-activated receptor 1 (PAR-1) selective activating peptide. Biochem/physiol Actions

SF1126 is a water soluble, small-molecule prodrug containing the pan-PI3K/mTOR inhibitor LY294002/SF1101 conjugated to the RGD-containing tetra-peptide SF1174 with potential antineoplastic and antiangiogenic activities. The SF1126 is designed to

SF1126 is a water soluble, small-molecule prodrug containing the pan-PI3K/mTOR inhibitor LY294002/SF1101 conjugated to the RGD-containing tetra-peptide SF1174 with potential antineoplastic and antiangiogenic activities. The SF1126 is designed to

Biochem/physiol Actions SF3B1 Protein degrader (reported as PROTAC-O4I2 in Gama-Brambila et al.) is a cell permeable degrader of splicing factor 3B1 (SF3B1) containing an SF3B1 activator O4I2 connected to the ligand of the cereblon ubiquitin""

Biochem/physiol Actions SF3B1 Protein degrader (reported as PROTAC-O4I2 in Gama-Brambila et al.) is a cell permeable degrader of splicing factor 3B1 (SF3B1) containing an SF3B1 activator O4I2 connected to the ligand of the cereblon ubiquitin""

SG-Carboxypeptidase B (Recombinant)&tradeis the rat carboxypeptidase B expressed in E. coli.

SG-Carboxypeptidase B (Recombinant)&tradeis the rat carboxypeptidase B expressed in E. coli.

Shepherdin (79-87) TFA is amino acids 79 to 87 fragment of Shepherdin. Shepherdin is a peptidomimetic antagonist of the complex between Hsp90 and Survivin . Anticancer activity.Appearance:SolidBiological Activity:Shepherdin (79-87) TFA is amino

Shepherdin (79-87) TFA is amino acids 79 to 87 fragment of Shepherdin. Shepherdin is a peptidomimetic antagonist of the complex between Hsp90 and Survivin . Anticancer activity.Appearance:SolidBiological Activity:Shepherdin (79-87) TFA is amino