D-VAL-PHE-LYS CHLOROMETHYL K 1PC X 5MG (C005B-231444)

General description

Selective irreversible inhibitor of plasmin with high selectivity for plasmin (IC₅₀ = 100 pM for human plasmin) over urokinase.

Selective irreversible inhibitor of plasmin with high selectivity for plasmin over urokinase.

Biochem/physiol Actions

Cell permeable: no

Primary Target
Human plasmin

Product does not compete with ATP.

Reversible: no

Target IC₅₀: 100 pM for human plasmin

Packaging

Packaged under inert gas

Warning

Toxicity: Standard Handling (A)

Sequence

H-D-Val-Phe-Lys-CMK

Reconstitution

Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 1 month at -20°C.







From Catalog:

Desc. Field- added "(IC₅₀ = 100 pM for human plasmin) "

Other Notes

Woessner, J.F., Jr., et al. 1989. Steroids54, 491.

Legal Information

CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany

Quality Level: 100. Assay: ≥. 90% (TLC). form: lyophilized solid. manufacturer/tradename: Calbiochem^®. . storage condition: OK to freeze, desiccated. color: off-white. solubility: DMSO: 5 . mg/mL. shipped in: ambient. storage temp.: 2-8°C. Storage Class Code: 11 - Combustible Solids. WGK: WGK 1. Flash Point(F): Not applicable. Flash Point(C): Not applicable.