DCLX069 is a selective protein arginine methyltransferase 1 (PRMT1) inhibitor with an IC 50 value of 17.9 µM. DCLX069 shows less active against PRMT4 and PRMT6 . DCLX069 has anticancer effectsIn VitroDCLX069 (12.5-100 µM) effectively blocks cell proliferation in breast cancer, liver cancer and acute myeloid leukemia cell lines (MCF7, HepG2, and THP1 cells) in a concentration-dependent manner. MCE has not independently confirmed the accuracy of these methods. They are for reference only.Form:SolidIC50& Target:PRMT1 17.9 μM (IC 50 ). Specification: 0.98 Molecular Formula: C20H25N3O2 Molecular Weight: 339.43
- UPC:
- 12352005
- Condition:
- New
- Availability:
- 8-12 weeks
- Weight:
- 1.06 Ounces
- HazmatClass:
- No
- WeightUOM:
- LB
- MPN:
- D650930-100mg
- CAS:
- 792946-69-1
- Product Size:
- 100mg
