General description
A potent agonist selective for δ opioid receptor (EC50 = 5.2 nM). Exhibits anti-convulsant effects in vivo in rats, also used in nociceptive studies.
Biochem/physiol Actions
Primary Target
δ opioid receptor
Warning
Toxicity: Standard Handling (A)
Sequence
Tyr-D-Pen-Gly-Phe-D-Pen (2-5 disulfide bond)
Reconstitution
Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
Other Notes
Chen, C., 1997. J. Pharmacol. Exp. Ther.283, 1151.
Chandrakumar, S., et al., 1992. J. Med. Chem.35, 2928.
Tortella, F. 1988. Peptides.9, 1177.
Clark, A., et al., 1986. Eur. J. Pharmacol.128, 303.
Legal Information
CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany
- UPC:
- 51152023
- Condition:
- New
- Weight:
- 1.00 Ounces
- HazmatClass:
- No
- WeightUOM:
- LB
- MPN:
- 5081600001
