Tyrosine kinase inhibitors

PrEST Antigen CDKN2B cyclin-dependent kinase inhibitor 2B (p

PrEST Antigen CDKN2C cyclin-dependent kinase inhibitor 2C (p

Synonym(s): Leu-Ser-Glu-Thr-Lys-Pro-Ala-Val Formula: C37H65N9O13 Formula weight: 843.98 Harmonized Tariff Code:  2933.99

Synonym(s): K252a Formula: C27H21N3O5 Formula weight: 467.47 CAS Number: 97161-97-2 Harmonized Tariff Code:  2933.29

A convenient set that offers several highly selective serine/threonine kinase inhibitors. Kinases play an important role in numerous signaling cascades.

A cell-permeable pyrazolocarbohydrazide compound that acts as a potent, reversible, sphingosine competitive and ATP-non-competitive inhibitor of sphingosine kinase 1 (SphK1) activity with excellent selectivity over SphK2 (K i = 1.33 and &gt&gt25

A cell-permeable imidazopyrimidine compound that acts a potent, ATP-competitive, reversible, and highly selective inhibitor of Syk tyrosine kinase activity (IC 50 = 10 nM) with no inhibitory effect against Btk, Fyn, Itk, Lyn, and Src even at

A cell-permeable, bioactive, non-toxic quinoline based compound that acts as a highly potent, ATP-non-competitive, tight-binding type II TAM (Tyro3, Axl, and Mer) kinase inhibitor (IC 50 = 8, 29, and 5 nM, respectively for Tyro3, Axl, and Mer).

GenScript Tyrosine Protein Kinase JAK 2 (Phospho-Tyr 8, 9 ) is a peptide corresponding to amino acids 475 to 491 of mouse JAK2, a member of the Janus kinase (Jak) family of cytoplasmic protein tyrosine kinases.

A cell-permeable 3-substituted indolin-2-one compound that acts as a reversible and ATP-competitive VEGF receptor tyrosine kinase inhibitor. At low concentration (&#88045 &#181M), it specifically blocks VEGF-C- (Cat.