Edonentan (BMS 207940) is an antagonist for endothelin receptor ( ET A receptor ), with a K i of 10 pM. Edonentan is metabolic stable, exhibits good pharmakokinetic characters in rats. Edonentan regulates the endothelin system, blocks the big Endothelin-induced pressor response in rats model .
Molecular Formula: C28H32N4O5S
Molecular Weight: 536.64
PubChem CID: 156690
Isomeric SMILES: CC1=C(ON=C1NS(=O)(=O)C2=CC=CC=C2C3=C(C=C(C=C3)C4=NC=CO4)CN(C)C(=O)CC(C)(C)C)C
- UPC:
- 51172905
- Condition:
- New
- Availability:
- 4-8 weeks
- Weight:
- 1.06 Ounces
- HazmatClass:
- No
- WeightUOM:
- LB
- MPN:
- E1362910-1mg
- Product Size:
- 1mg
- CAS:
- 210891-04-6