General description
An irreversible inhibitor of urokinase (IC50<1 µM) and Factor Xa.
Biochem/physiol Actions
Cell permeable: no
Primary Target
urokinase
Product does not compete with ATP.
Reversible: no
Target IC50: <1 µM against urokinase
Warning
Toxicity: Standard Handling (A)
Sequence
H-Glu-Gly-Arg-CMK
Reconstitution
Following reconstitution aliquot and freeze (-20°C). Stock solutions are stable for up to 1 month at -20°C. Avoid freeze/thaw cycles of stock solution.
Other Notes
Kettner, C., and Shaw, E. 1979. Biochim. Biophys. Acta569, 31.
Legal Information
CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany
Molecular Weight: 392.84. Empirical Formula: C14H25ClN6O5. Quality Level: 100. Assay: ≥. 80% (HPLC). form: solid. manufacturer/tradename: Calbiochem®. . storage condition: OK to freeze, desiccated (hygroscopic). color: white. solubility: water: 50 . mg/mL. shipped in: ambient. storage temp.: −. 20°C. Storage Class Code: 11 - Combustible Solids. WGK: WGK 1. Flash Point(F): Not applicable. Flash Point(C): Not applicable.- UPC:
- 41116133
- Condition:
- New
- Weight:
- 1.00 Ounces
- HazmatClass:
- No
- WeightUOM:
- LB
- MPN:
- 347436-5MG