A potent inhibitor of PORCN (EC50 = 0.5 nM); displays high stability in human plasma (t1/2 > 24 hours) and in zebrafish, but is much less stable in plasma from mice and rats; completely blocks Wnt/β-catenin-dependent developmental processes in zebrafish and in cultured mouse embryonic kidneys.
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- UPC:
- 51172832
- Condition:
- New
- Availability:
- 3 Days
- Weight:
- 1.00 Ounces
- HazmatClass:
- No
- WeightUOM:
- LB
- MPN:
- 15243-10
- Model Number:
- C818F76
- Temperature Control Device:
- Yes