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90052-50A structural analog of capsaicin with complex interactions in the CB system inhibits the reuptake of AEA, acts as CB1 receptor agonist and is resistant to FAAH hydrolysis exhibits vasodilator, analgesic, and anti-inflammatory properties.
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13622-10A potent inhibitor of PI3K with selectivity for the class IB isoform PI3K&gamma (IC<sub>50</sub> = 70 nM), compared to PI3K&alpha (IC<sub>50</sub> = 240 nM), PI3K&beta (IC<sub>50</sub> = 1.45 &muM), and PI3K&delta (IC<sub>50</sub> =1.
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13622-25A potent inhibitor of PI3K with selectivity for the class IB isoform PI3K&gamma (IC<sub>50</sub> = 70 nM), compared to PI3K&alpha (IC<sub>50</sub> = 240 nM), PI3K&beta (IC<sub>50</sub> = 1.45 &muM), and PI3K&delta (IC<sub>50</sub> =1.
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13622-5A potent inhibitor of PI3K with selectivity for the class IB isoform PI3K&gamma (IC<sub>50</sub> = 70 nM), compared to PI3K&alpha (IC<sub>50</sub> = 240 nM), PI3K&beta (IC<sub>50</sub> = 1.45 &muM), and PI3K&delta (IC<sub>50</sub> =1.
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13622-50A potent inhibitor of PI3K with selectivity for the class IB isoform PI3K&gamma (IC<sub>50</sub> = 70 nM), compared to PI3K&alpha (IC<sub>50</sub> = 240 nM), PI3K&beta (IC<sub>50</sub> = 1.45 &muM), and PI3K&delta (IC<sub>50</sub> =1.
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10626-1An agonist of GPR199 that is effective both in isolated cells and in vivo increases cAMP levels in HEK293 cells transfected with human GPR119 (EC50 = 2.5 &muM) and promotes glucose-stimulated insulin secretion in mice (100 mg/kg).
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10626-10An agonist of GPR199 that is effective both in isolated cells and in vivo increases cAMP levels in HEK293 cells transfected with human GPR119 (EC50 = 2.5 &muM) and promotes glucose-stimulated insulin secretion in mice (100 mg/kg).
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10626-25An agonist of GPR199 that is effective both in isolated cells and in vivo increases cAMP levels in HEK293 cells transfected with human GPR119 (EC50 = 2.5 &muM) and promotes glucose-stimulated insulin secretion in mice (100 mg/kg).
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10626-5An agonist of GPR199 that is effective both in isolated cells and in vivo increases cAMP levels in HEK293 cells transfected with human GPR119 (EC50 = 2.5 &muM) and promotes glucose-stimulated insulin secretion in mice (100 mg/kg).
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14978-1Formal Name: N-[(1S)-2-hydroxy-1-phenylethyl]-N'-[4-(4-pyridinyl)phenyl]-urea CAS Number: 928320-12-1 Molecular Formula: C<sub>20</sub>H<sub>19</sub>N<sub>3</sub>O<sub>2</sub>
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14978-10Formal Name: N-[(1S)-2-hydroxy-1-phenylethyl]-N'-[4-(4-pyridinyl)phenyl]-urea CAS Number: 928320-12-1 Molecular Formula: C<sub>20</sub>H<sub>19</sub>N<sub>3</sub>O<sub>2</sub>
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14978-25Formal Name: N-[(1S)-2-hydroxy-1-phenylethyl]-N'-[4-(4-pyridinyl)phenyl]-urea CAS Number: 928320-12-1 Molecular Formula: C<sub>20</sub>H<sub>19</sub>N<sub>3</sub>O<sub>2</sub>