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13307-25A competitive inhibitor of PC-PLC (Ki = 6.4 µM) also reduces sphingomyelin synthase activity, both in membrane preparations (IC<sub>50</sub> = 100 µg/ml) and in cells has antioxidant, antiviral, and anti-tumor activities.
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13307-5A competitive inhibitor of PC-PLC (Ki = 6.4 µM) also reduces sphingomyelin synthase activity, both in membrane preparations (IC<sub>50</sub> = 100 µg/ml) and in cells has antioxidant, antiviral, and anti-tumor activities.
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17282-1A Cdc25 phosphatase inhibitor (IC<sub>50</sub> = 0.82 µM for human recombinant Cdc25B) arrests asynchronous PC-3 prostate cancer cells in G2/M phase at 20 µM.
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17282-10A Cdc25 phosphatase inhibitor (IC<sub>50</sub> = 0.82 µM for human recombinant Cdc25B) arrests asynchronous PC-3 prostate cancer cells in G2/M phase at 20 µM.
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17282-25A Cdc25 phosphatase inhibitor (IC<sub>50</sub> = 0.82 µM for human recombinant Cdc25B) arrests asynchronous PC-3 prostate cancer cells in G2/M phase at 20 µM.
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17282-5A Cdc25 phosphatase inhibitor (IC<sub>50</sub> = 0.82 µM for human recombinant Cdc25B) arrests asynchronous PC-3 prostate cancer cells in G2/M phase at 20 µM.
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17131-10A double prodrug that undergoes in vivo hydrolytic cleavage to produce dabigatran, a potent thrombin inhibitor (Ki = 4.5 nM) shows antithrombotic efficacy in animal models of thrombosis, with a rapid onset of action.
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17131-5A double prodrug that undergoes in vivo hydrolytic cleavage to produce dabigatran, a potent thrombin inhibitor (Ki = 4.5 nM) shows antithrombotic efficacy in animal models of thrombosis, with a rapid onset of action.
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17131-50A double prodrug that undergoes in vivo hydrolytic cleavage to produce dabigatran, a potent thrombin inhibitor (Ki = 4.5 nM) shows antithrombotic efficacy in animal models of thrombosis, with a rapid onset of action.
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18451-1Molecular Formula: C<sub>24</sub>H<sub>28</sub>D<sub>13</sub>N<sub>7</sub>O<sub>5</sub> Formula Weight: 640.8
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18451-500Molecular Formula: C<sub>24</sub>H<sub>28</sub>D<sub>13</sub>N<sub>7</sub>O<sub>5</sub> Formula Weight: 640.8
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17133-1A potent thrombin inhibitor (Ki = 4.5 nM) also inhibits trypsin (Ki = 50.3 nM), but only weakly inhibits other serine proteases has poor bioavailability after oral administration.