-
10005223-10A selective inhibitor of AEA uptake that is resistant to FAAH hydrolysis is the structurally "reversed" isomer of AM404 blocks the uptake of tritiated AEA with an EC50 value of about 1.5 µM in mouse cortical neurons.
-
10005223-100A selective inhibitor of AEA uptake that is resistant to FAAH hydrolysis is the structurally "reversed" isomer of AM404 blocks the uptake of tritiated AEA with an EC50 value of about 1.5 µM in mouse cortical neurons.
-
10005223-5A selective inhibitor of AEA uptake that is resistant to FAAH hydrolysis is the structurally "reversed" isomer of AM404 blocks the uptake of tritiated AEA with an EC50 value of about 1.5 µM in mouse cortical neurons.
-
10005223-50A selective inhibitor of AEA uptake that is resistant to FAAH hydrolysis is the structurally "reversed" isomer of AM404 blocks the uptake of tritiated AEA with an EC50 value of about 1.5 µM in mouse cortical neurons.
-
10006972-1A potent and selective CB1 receptor antagonist/inverse agonist (Ki = 12 and 4,200 nM for CB1 and CB2, respectively)
-
10006972-10A potent and selective CB1 receptor antagonist/inverse agonist (Ki = 12 and 4,200 nM for CB1 and CB2, respectively)
-
10006972-5A potent and selective CB1 receptor antagonist/inverse agonist (Ki = 12 and 4,200 nM for CB1 and CB2, respectively)
-
90060-10An analog of AEA that potentiates the activity of endogenous AEA by blocking its re-uptake into presynaptic neurons selectively inhibits the carrier-mediated transport of AEA without affecting anandamide hydrolysis inhibits the transport of AEA
-
90060-100An analog of AEA that potentiates the activity of endogenous AEA by blocking its re-uptake into presynaptic neurons selectively inhibits the carrier-mediated transport of AEA without affecting anandamide hydrolysis inhibits the transport of AEA
-
90060-5An analog of AEA that potentiates the activity of endogenous AEA by blocking its re-uptake into presynaptic neurons selectively inhibits the carrier-mediated transport of AEA without affecting anandamide hydrolysis inhibits the transport of AEA
-
90060-50An analog of AEA that potentiates the activity of endogenous AEA by blocking its re-uptake into presynaptic neurons selectively inhibits the carrier-mediated transport of AEA without affecting anandamide hydrolysis inhibits the transport of AEA
-
15261-1A retinoic acid receptor agonist that is selective for RAR&alpha (Kd = 8 nM AC50 = 0.36 nM) compared to RAR&beta (Kd = 131 nM AC50 = 24.