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18227-1A corticosteroid prodrug that is converted to its active form, des-CIC, a glucocorticoid receptor agonist (Ki = 0.31 nM) used to ameliorate symptoms of airway inflammatory diseases.
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18227-10A corticosteroid prodrug that is converted to its active form, des-CIC, a glucocorticoid receptor agonist (Ki = 0.31 nM) used to ameliorate symptoms of airway inflammatory diseases.
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18227-5A corticosteroid prodrug that is converted to its active form, des-CIC, a glucocorticoid receptor agonist (Ki = 0.31 nM) used to ameliorate symptoms of airway inflammatory diseases.
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18227-50A corticosteroid prodrug that is converted to its active form, des-CIC, a glucocorticoid receptor agonist (Ki = 0.31 nM) used to ameliorate symptoms of airway inflammatory diseases.
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15194-1A competitive inhibitor of nucleotide binding by Ras-related GTPases binds Rab7 (Ki = 13 nM), preventing BODIPY-linked GTP and GDP binding with EC<sub>50</sub> values of 11.2 and 21 nM, respectively.
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15194-10A competitive inhibitor of nucleotide binding by Ras-related GTPases binds Rab7 (Ki = 13 nM), preventing BODIPY-linked GTP and GDP binding with EC<sub>50</sub> values of 11.2 and 21 nM, respectively.
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15194-25A competitive inhibitor of nucleotide binding by Ras-related GTPases binds Rab7 (Ki = 13 nM), preventing BODIPY-linked GTP and GDP binding with EC<sub>50</sub> values of 11.2 and 21 nM, respectively.
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15194-5A competitive inhibitor of nucleotide binding by Ras-related GTPases binds Rab7 (Ki = 13 nM), preventing BODIPY-linked GTP and GDP binding with EC<sub>50</sub> values of 11.2 and 21 nM, respectively.
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15317-10An inhibitor of all three PKD isoforms (IC<sub>50</sub>s = 3.2, 0.
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15317-25An inhibitor of all three PKD isoforms (IC<sub>50</sub>s = 3.2, 0.
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15317-5An inhibitor of all three PKD isoforms (IC<sub>50</sub>s = 3.2, 0.
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12046-10A reversible, competitive antagonist of GPR35, blocking activation by the synthetic agonist pamoic acid with a Ki of 12.8 nM less potently blocks activation of GPR35 by zaprinast (IC50 = 160 nM) shows ~57-fold selectivity for GPR35 over the