Biologically Active Small Molecules

A synthetic version of the endogenous antidiuretic hormone arginine vasopressin acts as an agonist at human vasopressin V1a, V1b, and V2 receptors with Ki values of 62.4, 5.8, and 23.3 nM, respectively.

A synthetic version of the endogenous antidiuretic hormone arginine vasopressin acts as an agonist at human vasopressin V1a, V1b, and V2 receptors with Ki values of 62.4, 5.8, and 23.3 nM, respectively.

A synthetic version of the endogenous antidiuretic hormone arginine vasopressin acts as an agonist at human vasopressin V1a, V1b, and V2 receptors with Ki values of 62.4, 5.8, and 23.3 nM, respectively.

A cyclic hexadepsipeptide mycotoxin that has insecticidal activity.

A cyclic hexadepsipeptide mycotoxin that has insecticidal and phytotoxic activity induces apoptosis in human NSCLC cells.

DETA NONOate is a NO donor. It spontaneously dissociates in a pH-dependent, first-order process with a half-life of 20 hours and 56 hours at 37&degC and 22-25&degC, pH 7.4, respectively, to liberate 2 moles of NO per mole of parent compound.

DETA NONOate is a NO donor. It spontaneously dissociates in a pH-dependent, first-order process with a half-life of 20 hours and 56 hours at 37&degC and 22-25&degC, pH 7.4, respectively, to liberate 2 moles of NO per mole of parent compound.

DETA NONOate is a NO donor. It spontaneously dissociates in a pH-dependent, first-order process with a half-life of 20 hours and 56 hours at 37&degC and 22-25&degC, pH 7.4, respectively, to liberate 2 moles of NO per mole of parent compound.

DETA NONOate is a NO donor. It spontaneously dissociates in a pH-dependent, first-order process with a half-life of 20 hours and 56 hours at 37&degC and 22-25&degC, pH 7.4, respectively, to liberate 2 moles of NO per mole of parent compound.

A selective &alpha2-adrenoceptor agonist (Ki = 1.62 nM) that binds to &alpha1-adrenoceptors with much weaker potency (Ki = 415 nM) primarily used as a sedative for horses in large animal veterinary medicine.

A selective &alpha2-adrenoceptor agonist (Ki = 1.62 nM) that binds to &alpha1-adrenoceptors with much weaker potency (Ki = 415 nM) primarily used as a sedative for horses in large animal veterinary medicine.

A selective &alpha2-adrenoceptor agonist (Ki = 1.62 nM) that binds to &alpha1-adrenoceptors with much weaker potency (Ki = 415 nM) primarily used as a sedative for horses in large animal veterinary medicine.