ligands acting on targets

Product Describtion:JQ1 is a member of the triazolo-diazepine compound family, which functions as a pan-BET (bromodomain and extra-terminal motif) family inhibitor. JQ1 is known to suppress cell proliferation and therefore, can be used as a

Product Describtion:JQ1 is a member of the triazolo-diazepine compound family, which functions as a pan-BET (bromodomain and extra-terminal motif) family inhibitor. JQ1 is known to suppress cell proliferation and therefore, can be used as a

Product Describtion:JQ1 is a member of the triazolo-diazepine compound family, which functions as a pan-BET (bromodomain and extra-terminal motif) family inhibitor. JQ1 is known to suppress cell proliferation and therefore, can be used as a

Product Describtion:JQ1 is a member of the triazolo-diazepine compound family, which functions as a pan-BET (bromodomain and extra-terminal motif) family inhibitor. JQ1 is known to suppress cell proliferation and therefore, can be used as a

Information(+)-JQ1 is a BET bromodomain inhibitor, with IC50 of 77 nM/33 nM for BRD4(1/2) in cell-free assays, binding to all bromodomains of the BET family, but not to bromodomains outside the BET family. (+)-JQ1 suppresses cell proliferation via

(+)-JQ1 carboxylic acid.

(+)-JQ1 carboxylic acid.

(+)-JQ1 carboxylic acid.

(+)-JQ1 carboxylic acid.

Functionalized BET bromodomain inhibitor: 'click' target ligand for PROTACs.

Functionalized BET bromodomain inhibitor: 'click' target ligand for PROTACs.

Functionalized BET bromodomain inhibitor: 'click' target ligand for PROTACs.