ligands acting on targets

(R,R)-CXCR2-IN-2, diastereoisomer of CXCR2-IN-2 (compound 68), is a brain penetrant CXCR2 antagonist with a pIC 50 of 9 and 6.8 in the Tango assay and d in the HWB Gro-α induced CD11b expression assay, respectively.Form:Solid.

(R,R)-CXCR2-IN-2, diastereoisomer of CXCR2-IN-2 (compound 68), is a brain penetrant CXCR2 antagonist with a pIC 50 of 9 and 6.8 in the Tango assay and d in the HWB Gro-α induced CD11b expression assay, respectively.

Formoterol(Arformoterol) is a novel highly β2-selective adrenergic agonist and holds promise as a β 2-agonist that could impart selective beneficial metabolic effects.

Formoterol(Arformoterol) is a novel highly β2-selective adrenergic agonist and holds promise as a β 2-agonist that could impart selective beneficial metabolic effects.

(R,R)-GSK321 is a wild-type isocitrate dehydrogenase 1 ( WT IDH1 ) inhibitor with an IC 50 value of 120 nM. (R,R)-GSK321 as a mutant R132H IDH1 inhibitor, is an isomer of GSK321 with some wild-type cross reactivityIn Vitro(R,R)-GSK321 (0.1~3 μM: 5

(R,R)-GSK321 is a wild-type isocitrate dehydrogenase 1 ( WT IDH1 ) inhibitor with an IC 50 value of 120 nM. (R,R)-GSK321 as a mutant R132H IDH1 inhibitor, is an isomer of GSK321 with some wild-type cross reactivityIn Vitro(R,R)-GSK321 (0.1~3 μM: 5

(R,R)-Labetalol is a competitive antagonist at both α-AR and β-AR (α-and β-adrenergic receptor) sites.

Potent subtype-selective ligand: ERα agonist/ERβ antagonist.

(R,R)-VVD-118313 is the isomer of VVD-118313 ( HY-151385 ). VVD-118313 is a selective JAK1 inhibitor and blocks JAK1-dependent trans-phosphorylation and cytokine signaling. VVD-118313 can be used for research of cancerIn VitroVVD-118313 (compound

(R,R)-VVD-118313 is the isomer of VVD-118313 ( HY-151385 ). VVD-118313 is a selective JAK1 inhibitor and blocks JAK1-dependent trans-phosphorylation and cytokine signaling. VVD-118313 can be used for research of cancerIn VitroVVD-118313 (compound

(R,R)-VVD-118313 is the isomer of VVD-118313 ( HY-151385 ). VVD-118313 is a selective JAK1 inhibitor and blocks JAK1-dependent trans-phosphorylation and cytokine signaling. VVD-118313 can be used for research of cancerIn VitroVVD-118313 (compound

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