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G654663-1mlGAT211 is a cannabinoid 1 receptor (CB1R) positive allosteric modulator (PAM). GAT211 activates cAMP and β-arrestin2 with EC 50 values of 260 nM and 650 nM, respectively. GAT211 inhibits GAT211 can be used for neuropathic and/or inflammatory pain
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G659189-100mgGB-110 hydrochloride is a potent, orally active, and nonpeptidic protease activated receptor 2 (PAR2) agonist. GB-110 hydrochloride selectively induces PAR2-mediated intracellular Ca 2+ release in HT29 cells with an EC 50 of 0.28
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G659189-10mgGB-110 hydrochloride is a potent, orally active, and nonpeptidic protease activated receptor 2 (PAR2) agonist. GB-110 hydrochloride selectively induces PAR2-mediated intracellular Ca 2+ release in HT29 cells with an EC 50 of 0.28
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G659189-25mgGB-110 hydrochloride is a potent, orally active, and nonpeptidic protease activated receptor 2 (PAR2) agonist. GB-110 hydrochloride selectively induces PAR2-mediated intracellular Ca 2+ release in HT29 cells with an EC 50 of 0.28
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G659189-50mgGB-110 hydrochloride is a potent, orally active, and nonpeptidic protease activated receptor 2 (PAR2) agonist. GB-110 hydrochloride selectively induces PAR2-mediated intracellular Ca 2+ release in HT29 cells with an EC 50 of 0.28
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G659189-5mgGB-110 hydrochloride is a potent, orally active, and nonpeptidic protease activated receptor 2 (PAR2) agonist. GB-110 hydrochloride selectively induces PAR2-mediated intracellular Ca 2+ release in HT29 cells with an EC 50 of 0.28
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G661669-1mlGB-110 hydrochloride is a potent, orally active, and nonpeptidic protease activated receptor 2 (PAR2) agonist. GB-110 hydrochloride selectively induces PAR2-mediated intracellular Ca 2+ release in HT29 cells with an EC 50 of 0.28 μM.IC50&:
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G649297-100mgGCN2-IN-1 (A-92) is a potent general control nonderepressible 2 kinase ( GCN2 ) inhibitor with an IC 50 of <:0.3 μM in the enzyme assay and an IC 50 of 0.3-3 μM in the cell assayIn VitroGCN2-IN-1 (Compound A-92) is a GCN2 inhibitor, which may be
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G649297-10mgGCN2-IN-1 (A-92) is a potent general control nonderepressible 2 kinase ( GCN2 ) inhibitor with an IC 50 of <:0.3 μM in the enzyme assay and an IC 50 of 0.3-3 μM in the cell assayIn VitroGCN2-IN-1 (Compound A-92) is a GCN2 inhibitor, which may be
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G649297-1mgGCN2-IN-1 (A-92) is a potent general control nonderepressible 2 kinase ( GCN2 ) inhibitor with an IC 50 of <:0.3 μM in the enzyme assay and an IC 50 of 0.3-3 μM in the cell assayIn VitroGCN2-IN-1 (Compound A-92) is a GCN2 inhibitor, which may be
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G649297-25mgGCN2-IN-1 (A-92) is a potent general control nonderepressible 2 kinase ( GCN2 ) inhibitor with an IC 50 of <:0.3 μM in the enzyme assay and an IC 50 of 0.3-3 μM in the cell assayIn VitroGCN2-IN-1 (Compound A-92) is a GCN2 inhibitor, which may be
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G649297-50mgGCN2-IN-1 (A-92) is a potent general control nonderepressible 2 kinase ( GCN2 ) inhibitor with an IC 50 of <:0.3 μM in the enzyme assay and an IC 50 of 0.3-3 μM in the cell assayIn VitroGCN2-IN-1 (Compound A-92) is a GCN2 inhibitor, which may be