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G649529-25mgGS-626510 is a potent, and orally active BET family bromodomains inhibitor, with K d values of 0.59-3.2 nM for BRD2/3/4, with IC 50 values of 83 nM and 78 nM foe BD1 and BD2 , respectivelyForm:SolidIC50&: Target:BRD2 0.59-2.5 nM (Kd) BRD3
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G649529-50mgGS-626510 is a potent, and orally active BET family bromodomains inhibitor, with K d values of 0.59-3.2 nM for BRD2/3/4, with IC 50 values of 83 nM and 78 nM foe BD1 and BD2 , respectivelyForm:SolidIC50&: Target:BRD2 0.59-2.5 nM (Kd) BRD3
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G649529-5mgGS-626510 is a potent, and orally active BET family bromodomains inhibitor, with K d values of 0.59-3.2 nM for BRD2/3/4, with IC 50 values of 83 nM and 78 nM foe BD1 and BD2 , respectivelyForm:SolidIC50&: Target:BRD2 0.59-2.5 nM (Kd) BRD3
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G655895-1mlGS-626510 is a potent, and orally active BET family bromodomains inhibitor, with K d values of 0.59-3.2 nM for BRD2/3/4, with IC 50 values of 83 nM and 78 nM foe BD1 and BD2 , respectivelyIC50&: Target:BRD2 0.59-2.5 nM (Kd) BRD3 0.65-0.66 nM (Kd)
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G659015-10mgGSK 690 (Hydrochloride) is a reversible inhibitor of lysine specific demethylase 1 (LSD1) , with a K d value of 9 nM and a biochemical IC 50 of 37 nM.Appearance:SolidIC50&: Target:IC50: 37 nM (LSD1), Kd: 8 nM (LSD1) .In Vitro:GSK690 (1-10 μM)
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G659015-25mgGSK 690 (Hydrochloride) is a reversible inhibitor of lysine specific demethylase 1 (LSD1) , with a K d value of 9 nM and a biochemical IC 50 of 37 nM.Appearance:SolidIC50&: Target:IC50: 37 nM (LSD1), Kd: 8 nM (LSD1) .In Vitro:GSK690 (1-10 μM)
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G659015-50mgGSK 690 (Hydrochloride) is a reversible inhibitor of lysine specific demethylase 1 (LSD1) , with a K d value of 9 nM and a biochemical IC 50 of 37 nM.Appearance:SolidIC50&: Target:IC50: 37 nM (LSD1), Kd: 8 nM (LSD1) .In Vitro:GSK690 (1-10 μM)
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G659015-5mgGSK 690 (Hydrochloride) is a reversible inhibitor of lysine specific demethylase 1 (LSD1) , with a K d value of 9 nM and a biochemical IC 50 of 37 nM.Appearance:SolidIC50&: Target:IC50: 37 nM (LSD1), Kd: 8 nM (LSD1) .In Vitro:GSK690 (1-10 μM)
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G661638-1mlGSK 690 (Hydrochloride) is a reversible inhibitor of lysine specific demethylase 1 (LSD1) , with a K d value of 9 nM and a biochemical IC 50 of 37 nM.IC50&: Target:IC50: 37 nM (LSD1), Kd: 8 nM (LSD1) .In Vitro:GSK690 (1-10 μM) acts together with
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G651347-10mgGSK-269984A is a Prostaglandin E2 Receptor 1 (EP1) antagonist with a pIC 50 of 7.9.In VitroResults from [ 3 H]-PGE 2 binding assay in CHO cells overexpressing the human EP 1 receptor demonstrate that GSK-269984A is an antagonist of EP 1 receptor
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G651347-5mgGSK-269984A is a Prostaglandin E2 Receptor 1 (EP1) antagonist with a pIC 50 of 7.9.In VitroResults from [ 3 H]-PGE 2 binding assay in CHO cells overexpressing the human EP 1 receptor demonstrate that GSK-269984A is an antagonist of EP 1 receptor
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G658851-10mgGSK-2793660 is an orally active and irreversible inhibitor of Cathepsin C ( CTSC ). GSK-2793660 can be used for the research of bronchiectasis.Appearance:SolidIC50&: Target:Cathepsin C (CTSC)In Vivo:GSK-2793660 is a cathepsin C (also known as