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H648109-5mghCAII-IN-8, an amide, is a highly selective carbonic anhydrase (CA) inhibitor with an IC 50 value of 0.18 μM against hCA IIIn VitrohCAII-IN-8 (compound 9: 100 μM: 24-48 h) has noncytotoxic on HEK-293 T cells (cell viability>:90%) compared to the
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H646786-100mgHCV-IN-30 (compound 48) is a HCV NS5A replication complex inhibitor, with IC 50 s of 901 and 102 nM for genotypes 1a and 1b replicons, respectively.Form:Solid.
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H646786-25mgHCV-IN-30 (compound 48) is a HCV NS5A replication complex inhibitor, with IC 50 s of 901 and 102 nM for genotypes 1a and 1b replicons, respectively.Form:Solid.
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H646786-50mgHCV-IN-30 (compound 48) is a HCV NS5A replication complex inhibitor, with IC 50 s of 901 and 102 nM for genotypes 1a and 1b replicons, respectively.Form:Solid.
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H650232-100mgHCV-IN-31 (compound 4) is a HCV inhibitor, with an EC 50 /EC 95 of 15.7 μM for HCV repliconForm:SolidIC50&: Target:EC50/EC95: 15.7 μM (HCV replicon).
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H650232-10mgHCV-IN-31 (compound 4) is a HCV inhibitor, with an EC 50 /EC 95 of 15.7 μM for HCV repliconForm:SolidIC50&: Target:EC50/EC95: 15.7 μM (HCV replicon).
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H650232-25mgHCV-IN-31 (compound 4) is a HCV inhibitor, with an EC 50 /EC 95 of 15.7 μM for HCV repliconForm:SolidIC50&: Target:EC50/EC95: 15.7 μM (HCV replicon).
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H650232-50mgHCV-IN-31 (compound 4) is a HCV inhibitor, with an EC 50 /EC 95 of 15.7 μM for HCV repliconForm:SolidIC50&: Target:EC50/EC95: 15.7 μM (HCV replicon).
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H650232-5mgHCV-IN-31 (compound 4) is a HCV inhibitor, with an EC 50 /EC 95 of 15.7 μM for HCV repliconForm:SolidIC50&: Target:EC50/EC95: 15.7 μM (HCV replicon).
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H656185-1mlHCV-IN-31 (compound 4) is a HCV inhibitor, with an EC 50 /EC 95 of 15.7 μM for HCV repliconIC50&: Target:EC50/EC95: 15.7 μM (HCV replicon).
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H649473-100mgHDAC-IN-4 is a selective HDAC6 and HDAC10 inhibitor with pIC 50 s of 7.2 and 6.8 in BRET assay, respectively. Antitumoral activityIn VitroHDAC-IN-4 inhibits HDAC1, HDAC2, HDAC3, HDAC8 and HDAC10 with pIC 50 s of 5.5, 4.6, 5.4, 5.4, 6.7 in FRET
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H649473-10mgHDAC-IN-4 is a selective HDAC6 and HDAC10 inhibitor with pIC 50 s of 7.2 and 6.8 in BRET assay, respectively. Antitumoral activityIn VitroHDAC-IN-4 inhibits HDAC1, HDAC2, HDAC3, HDAC8 and HDAC10 with pIC 50 s of 5.5, 4.6, 5.4, 5.4, 6.7 in FRET