Activin and Inhibin

Afizagabar (S44819) is a first-in-class, competitive, and selective antagonist at the GABA-binding site of the α5-GABAAR , with an IC 50 of 585 nM for α5β2γ2 and a K i of 66 nM for α5β3γ2. Afizagabar enhances hippocampal synaptic plasticity and

Afizagabar (S44819) is a first-in-class, competitive, and selective antagonist at the GABA-binding site of the α5-GABAAR , with an IC 50 of 585 nM for α5β2γ2 and a K i of 66 nM for α5β3γ2. Afizagabar enhances hippocampal synaptic plasticity and

Afizagabar (S44819) is a first-in-class, competitive, and selective antagonist at the GABA-binding site of the α5-GABAAR , with an IC 50 of 585 nM for α5β2γ2 and a K i of 66 nM for α5β3γ2. Afizagabar enhances hippocampal synaptic plasticity and

AFM-30a hydrochloride is a potent protein arginine deiminase 2 (PAD2) inhibitor and has excellent PAD2-selectivity. AFM-30a hydrochloride binds to PAD2 with an EC 50 value of 9.5 μM. AFM-30a hydrochloride also inhibits H3 citrullination with an EC

AFM-30a hydrochloride is a potent protein arginine deiminase 2 (PAD2) inhibitor and has excellent PAD2-selectivity. AFM-30a hydrochloride binds to PAD2 with an EC 50 value of 9.5 μM. AFM-30a hydrochloride also inhibits H3 citrullination with an EC

AFM-30a hydrochloride is a potent protein arginine deiminase 2 (PAD2) inhibitor and has excellent PAD2-selectivity. AFM-30a hydrochloride binds to PAD2 with an EC 50 value of 9.5 μM. AFM-30a hydrochloride also inhibits H3 citrullination with an EC

AG-09/1 is a specific formyl peptide receptor 1 ( FPR1 ) agonist. N-formyl peptide receptors (FPR) are important in host defenseIn VitroN-formyl peptides activate phagocytes through G protein-coupled receptors known as FPR. FPR1 was the first FPR

AG-09/1 is a specific formyl peptide receptor 1 ( FPR1 ) agonist. N-formyl peptide receptors (FPR) are important in host defenseIn VitroN-formyl peptides activate phagocytes through G protein-coupled receptors known as FPR. FPR1 was the first FPR

AG-09/1 is a specific formyl peptide receptor 1 ( FPR1 ) agonist. N-formyl peptide receptors (FPR) are important in host defenseIn VitroN-formyl peptides activate phagocytes through G protein-coupled receptors known as FPR. FPR1 was the first FPR

AG-09/1 is a specific formyl peptide receptor 1 ( FPR1 ) agonist. N-formyl peptide receptors (FPR) are important in host defenseIn VitroN-formyl peptides activate phagocytes through G protein-coupled receptors known as FPR. FPR1 was the first FPR

AG-09/1 is a specific formyl peptide receptor 1 ( FPR1 ) agonist. N-formyl peptide receptors (FPR) are important in host defenseIn VitroN-formyl peptides activate phagocytes through G protein-coupled receptors known as FPR. FPR1 was the first FPR

AG-270 is an allosteric, noncompetitive, first-in-class, reversible and orally active MAT2A inhibitor, with an IC 50 of 14 nMIn VitroAG-270 demonstrates potent reduction in levels of intracellular SAM , as well as MTAP-–selective antiproliferative