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A656905-1mlAGN 196996 is a potent and selective RARα antagonist with Ki value of 2 nM: little binding affinity for RARβ(Ki=1087 nM) and RARγ(Ki=8523 nM).IC50 value: 2 nM(Ki)Target: RARα antagonistAGN 196996 shows no activity in transactivation assays, but
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A646427-1mgAgomelatine-d 6 is deuterium labeled Agomelatine. Agomelatine is a specific agonist of MT1 and MT2 receptorsForm:SolidIC50&: Target:MT1, MT2.
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A646427-5mgAgomelatine-d 6 is deuterium labeled Agomelatine. Agomelatine is a specific agonist of MT1 and MT2 receptorsForm:SolidIC50&: Target:MT1, MT2.
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A650765-10mgAH3960 (compound 16c) is an antagonist of androgen receptor. AH3960 binds wild as well as T877 mutant type androgen receptors. AH3960 selectively inhibits T877 with an IC 50 value of 0.82 μM. AH3960 also serves as an agonist of parathyroid hormone
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A650765-25mgAH3960 (compound 16c) is an antagonist of androgen receptor. AH3960 binds wild as well as T877 mutant type androgen receptors. AH3960 selectively inhibits T877 with an IC 50 value of 0.82 μM. AH3960 also serves as an agonist of parathyroid hormone
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A650765-50mgAH3960 (compound 16c) is an antagonist of androgen receptor. AH3960 binds wild as well as T877 mutant type androgen receptors. AH3960 selectively inhibits T877 with an IC 50 value of 0.82 μM. AH3960 also serves as an agonist of parathyroid hormone
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A650765-5mgAH3960 (compound 16c) is an antagonist of androgen receptor. AH3960 binds wild as well as T877 mutant type androgen receptors. AH3960 selectively inhibits T877 with an IC 50 value of 0.82 μM. AH3960 also serves as an agonist of parathyroid hormone
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A651644-10mgAKB-6899, a prolyl hydroxylase domain 3 (PHD3) inhibitor, is a selective HIF-2α stabilizer. AKB-6899 also increases soluble form of the VEGF receptor (sVEGFR-1) production from GM-CSF-treated macrophages, and has antitumor and antiangiogenic
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A651644-25mgAKB-6899, a prolyl hydroxylase domain 3 (PHD3) inhibitor, is a selective HIF-2α stabilizer. AKB-6899 also increases soluble form of the VEGF receptor (sVEGFR-1) production from GM-CSF-treated macrophages, and has antitumor and antiangiogenic
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A651644-50mgAKB-6899, a prolyl hydroxylase domain 3 (PHD3) inhibitor, is a selective HIF-2α stabilizer. AKB-6899 also increases soluble form of the VEGF receptor (sVEGFR-1) production from GM-CSF-treated macrophages, and has antitumor and antiangiogenic
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A651644-5mgAKB-6899, a prolyl hydroxylase domain 3 (PHD3) inhibitor, is a selective HIF-2α stabilizer. AKB-6899 also increases soluble form of the VEGF receptor (sVEGFR-1) production from GM-CSF-treated macrophages, and has antitumor and antiangiogenic
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A656760-1mlAKB-6899, a prolyl hydroxylase domain 3 (PHD3) inhibitor, is a selective HIF-2α stabilizer. AKB-6899 also increases soluble form of the VEGF receptor (sVEGFR-1) production from GM-CSF-treated macrophages, and has antitumor and antiangiogenic