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A648011-5mgALDH1A1-IN-2 is a potent inhibitor of aldehyde dehydrogenase 1a1 ( aldh1a1 ). Aldehyde dehydrogenases (ALDH) constitute a family of enzymes that play a critical role in oxidizing various cytotoxic xenogenic and biogenic aldehydes. ALDH1A1-IN-2 has
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A648075-100mgALDH1A2-IN-1 is an active site-directed reversible ALDH1A2 inhibitor ( IC 50 =0.91 μM: Kd =0.26 μM) with several hydrophobic interactionsForm:SolidIC50&: Target:IC50: 0.91 μM (ALDH1A2), Kd: 0.26 μM (ALDH1A2).
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A648075-10mgALDH1A2-IN-1 is an active site-directed reversible ALDH1A2 inhibitor ( IC 50 =0.91 μM: Kd =0.26 μM) with several hydrophobic interactionsForm:SolidIC50&: Target:IC50: 0.91 μM (ALDH1A2), Kd: 0.26 μM (ALDH1A2).
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A648075-25mgALDH1A2-IN-1 is an active site-directed reversible ALDH1A2 inhibitor ( IC 50 =0.91 μM: Kd =0.26 μM) with several hydrophobic interactionsForm:SolidIC50&: Target:IC50: 0.91 μM (ALDH1A2), Kd: 0.26 μM (ALDH1A2).
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A648075-50mgALDH1A2-IN-1 is an active site-directed reversible ALDH1A2 inhibitor ( IC 50 =0.91 μM: Kd =0.26 μM) with several hydrophobic interactionsForm:SolidIC50&: Target:IC50: 0.91 μM (ALDH1A2), Kd: 0.26 μM (ALDH1A2).
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A648075-5mgALDH1A2-IN-1 is an active site-directed reversible ALDH1A2 inhibitor ( IC 50 =0.91 μM: Kd =0.26 μM) with several hydrophobic interactionsForm:SolidIC50&: Target:IC50: 0.91 μM (ALDH1A2), Kd: 0.26 μM (ALDH1A2).
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A655283-1mlALDH1A2-IN-1 is an active site-directed reversible ALDH1A2 inhibitor ( IC 50 =0.91 μM: Kd =0.26 μM) with several hydrophobic interactionsIC50&: Target:IC50: 0.91 μM (ALDH1A2), Kd: 0.26 μM (ALDH1A2).
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A648564-100mgALDH1A3-IN-1 (Compound 14) is a potent ALDH1A3 inhibitor, with an IC 50 of 0.63 µM and a K i of 0.46 µM. ALDH1A3-IN-1 can be studied in prostate cancerIn VitroALDH1A3-IN-1 (Compound 14) (0-200 µM, 96 h) shows antiproliferative activity in prostate
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A648564-10mgALDH1A3-IN-1 (Compound 14) is a potent ALDH1A3 inhibitor, with an IC 50 of 0.63 µM and a K i of 0.46 µM. ALDH1A3-IN-1 can be studied in prostate cancerIn VitroALDH1A3-IN-1 (Compound 14) (0-200 µM, 96 h) shows antiproliferative activity in prostate
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A648564-25mgALDH1A3-IN-1 (Compound 14) is a potent ALDH1A3 inhibitor, with an IC 50 of 0.63 µM and a K i of 0.46 µM. ALDH1A3-IN-1 can be studied in prostate cancerIn VitroALDH1A3-IN-1 (Compound 14) (0-200 µM, 96 h) shows antiproliferative activity in prostate
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A648564-50mgALDH1A3-IN-1 (Compound 14) is a potent ALDH1A3 inhibitor, with an IC 50 of 0.63 µM and a K i of 0.46 µM. ALDH1A3-IN-1 can be studied in prostate cancerIn VitroALDH1A3-IN-1 (Compound 14) (0-200 µM, 96 h) shows antiproliferative activity in prostate
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A648564-5mgALDH1A3-IN-1 (Compound 14) is a potent ALDH1A3 inhibitor, with an IC 50 of 0.63 µM and a K i of 0.46 µM. ALDH1A3-IN-1 can be studied in prostate cancerIn VitroALDH1A3-IN-1 (Compound 14) (0-200 µM, 96 h) shows antiproliferative activity in prostate