Approved Ligands

Argatroban is an anticoagulant that is a small molecule direct thrombin inhibitor.A peptidomimetic small molecule anticoagulant and direct thrombin inhibitor.

ARN-509 is a selective and competitive androgen receptor inhibitor with IC50 of 16 nM in a cell-free assay, useful for prostate cancer treatment.

ARN-509 is a selective and competitive androgen receptor inhibitor with IC50 of 16 nM in a cell-free assay, useful for prostate cancer treatment.

ARN-509 is a selective and competitive androgen receptor inhibitor with IC50 of 16 nM in a cell-free assay, useful for prostate cancer treatment.

Asenapine(Org 5222) inhibits adrenergic receptor (α1, α2A, α2B, α2C) with Ki of 0.25-1.2 nM and also inhibits 5-HT receptor (1A, 1B, 2A, 2B, 2C, 5A, 6, 7) with Ki of 0.03-4.0 nM.

Asenapine(Org 5222) inhibits adrenergic receptor (α1, α2A, α2B, α2C) with Ki of 0.25-1.2 nM and also inhibits 5-HT receptor (1A, 1B, 2A, 2B, 2C, 5A, 6, 7) with Ki of 0.03-4.0 nM.

Asenapine(Org 5222) inhibits adrenergic receptor (α1, α2A, α2B, α2C) with Ki of 0.25-1.2 nM and also inhibits 5-HT receptor (1A, 1B, 2A, 2B, 2C, 5A, 6, 7) with Ki of 0.03-4.0 nM.

Potent, selective histamine H1 receptor antagonist and potent hERG K + channel blocker.

Potent, selective histamine H1 receptor antagonist and potent hERG K + channel blocker.

Potent, selective histamine H1 receptor antagonist and potent hERG K + channel blocker.

(RS)-Atenolol is a cardioselective β-adrenergic blocker. It is considered to be antihypertensive, antianginal, and antiarrhythmic. (RS)-Atenolol is an inhibitor of β1-AR and β2-AR.An inhibitor of β1-AR and β2-AR.Atenolol is a β-adrenergic blocker

(RS)-Atenolol is a cardioselective β-adrenergic blocker. It is considered to be antihypertensive, antianginal, and antiarrhythmic. (RS)-Atenolol is an inhibitor of β1-AR and β2-AR.An inhibitor of β1-AR and β2-AR.Atenolol is a β-adrenergic blocker