Approved Ligands

Exendin-4 is an incretin mimetic peptide, which is composed of 39 amino acids. It is an analog of Glukagon-like peptide 1 (GLP-1), and an insulinotropic agent, with a long half-life. It was originally isolated from the venom of Gila monster lizard

InformationFadrozole (CGS16949A) Fadrozole (CGS16949A) is a potent, selective, nonsteroidal inhibitor of aromatase with an IC50 of 4.5 nM and selectivity over other cytochrome P-450 enzymes.TargetsAromatase 4.5 nM.

InformationFadrozole (CGS16949A) Fadrozole (CGS16949A) is a potent, selective, nonsteroidal inhibitor of aromatase with an IC50 of 4.5 nM and selectivity over other cytochrome P-450 enzymes.TargetsAromatase 4.5 nM.

InformationFadrozole (CGS16949A) Fadrozole (CGS16949A) is a potent, selective, nonsteroidal inhibitor of aromatase with an IC50 of 4.5 nM and selectivity over other cytochrome P-450 enzymes.TargetsAromatase 4.5 nM.

InformationFadrozole (CGS16949A) Fadrozole (CGS16949A) is a potent, selective, nonsteroidal inhibitor of aromatase with an IC50 of 4.5 nM and selectivity over other cytochrome P-450 enzymes.TargetsAromatase 4.5 nM.

InformationFadrozole (CGS16949A) Fadrozole (CGS16949A) is a potent, selective, nonsteroidal inhibitor of aromatase with an IC50 of 4.5 nM and selectivity over other cytochrome P-450 enzymes.TargetsAromatase 4.5 nM.

TG-101348 (SAR302503) is a selective inhibitor of JAK2 with IC50 of 3 nM, 35- and 334-fold more selective for JAK2 versus JAK1 and JAK3, TG-101348 also inhibit BRD4 with IC50 of 340 nM.A selective inhibitor of JAK2 tyrosine kinase.

TG-101348 (SAR302503) is a selective inhibitor of JAK2 with IC50 of 3 nM, 35- and 334-fold more selective for JAK2 versus JAK1 and JAK3, TG-101348 also inhibit BRD4 with IC50 of 340 nM.A selective inhibitor of JAK2 tyrosine kinase.

TG-101348 (SAR302503) is a selective inhibitor of JAK2 with IC50 of 3 nM, 35- and 334-fold more selective for JAK2 versus JAK1 and JAK3, TG-101348 also inhibit BRD4 with IC50 of 340 nM.A selective inhibitor of JAK2 tyrosine kinase.

Fenoldopam hydrochloride is a selective D1DR (D|1|-like dopamine receptor) partial agonist, a vasodilator, and also an AR (α|2|-adrenoceptor) antagonist|in vitro|. Fenoldopam hydrochloride does not readily cross the blood-brain barrier.

InformationFenoterol (Phenoterol) is aβ2 adrenoreceptoragonist with bronchodilator activity.Targetsβ2 adrenoreceptor.

InformationFenoterol (Phenoterol) is aβ2 adrenoreceptoragonist with bronchodilator activity.Targetsβ2 adrenoreceptor.