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A126115-5mgAG-1024 (Tyrphostin) inhibits IGF-1R autophosphorylation with IC50 of 7 μM, less potent to IR with IC50 of 57 μM.
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A125467-10mgAG14361 is a potent inhibitor of PARP1 with Ki of <:5 nM. It is at least 1000-fold more potent than the benzamides.
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A125467-50mgAG14361 is a potent inhibitor of PARP1 with Ki of <:5 nM. It is at least 1000-fold more potent than the benzamides.
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A125467-5mgAG14361 is a potent inhibitor of PARP1 with Ki of <:5 nM. It is at least 1000-fold more potent than the benzamides.