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A413448-100mgInformationAZ876 AZ876 is a novel high-affinity Liver X Receptor (LXR) agonist with Ki values of 0.007 μM and 0.011 μM for human LXRα and LXRβ respectively.TargetsLXRα : LXRβ 0.007 μM(Ki): 0.011 μM(Ki)In vitroIn binding assays, AZ876 is 25-fold and
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A413448-10mgInformationAZ876 AZ876 is a novel high-affinity Liver X Receptor (LXR) agonist with Ki values of 0.007 μM and 0.011 μM for human LXRα and LXRβ respectively.TargetsLXRα : LXRβ 0.007 μM(Ki): 0.011 μM(Ki)In vitroIn binding assays, AZ876 is 25-fold and
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A413448-1mgInformationAZ876 AZ876 is a novel high-affinity Liver X Receptor (LXR) agonist with Ki values of 0.007 μM and 0.011 μM for human LXRα and LXRβ respectively.TargetsLXRα : LXRβ 0.007 μM(Ki): 0.011 μM(Ki)In vitroIn binding assays, AZ876 is 25-fold and
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A413448-50mgInformationAZ876 AZ876 is a novel high-affinity Liver X Receptor (LXR) agonist with Ki values of 0.007 μM and 0.011 μM for human LXRα and LXRβ respectively.TargetsLXRα : LXRβ 0.007 μM(Ki): 0.011 μM(Ki)In vitroIn binding assays, AZ876 is 25-fold and
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A413448-5mgInformationAZ876 AZ876 is a novel high-affinity Liver X Receptor (LXR) agonist with Ki values of 0.007 μM and 0.011 μM for human LXRα and LXRβ respectively.TargetsLXRα : LXRβ 0.007 μM(Ki): 0.011 μM(Ki)In vitroIn binding assays, AZ876 is 25-fold and
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A607846-10mgAZ8838 is a potent, competitive, allosteric, orally active non-peptide small molecule antagonist of PAR2 with a pKi of 6.4 for hPAR2.
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A607846-1mgAZ8838 is a potent, competitive, allosteric, orally active non-peptide small molecule antagonist of PAR2 with a pKi of 6.4 for hPAR2.
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A607846-25mgAZ8838 is a potent, competitive, allosteric, orally active non-peptide small molecule antagonist of PAR2 with a pKi of 6.4 for hPAR2.
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A607846-5mgAZ8838 is a potent, competitive, allosteric, orally active non-peptide small molecule antagonist of PAR2 with a pKi of 6.4 for hPAR2.
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