Synthetic organic

EMD638683.

EMDT oxalate is a selective SR-6 agonist with a K|i|value of 16 nM. It activates adenylate cyclase at a comparable potency to serotonin.

EMDT oxalate is a selective SR-6 agonist with a K|i|value of 16 nM. It activates adenylate cyclase at a comparable potency to serotonin.

InformationEmedastine is a potent, high affinityhistamine H1-receptor-selectiveantagonist with Ki of 1.3 ±0.1 nM for H1-receptors while considerably weaker at H2- (K1 = 49,067 ± 11,113 nM) and H3-receptors (Ki = 12,430 ± 1,282 nM).TargetsH1 receptor

InformationEmedastine is a potent, high affinityhistamine H1-receptor-selectiveantagonist with Ki of 1.3 ±0.1 nM for H1-receptors while considerably weaker at H2- (K1 = 49,067 ± 11,113 nM) and H3-receptors (Ki = 12,430 ± 1,282 nM).TargetsH1 receptor

InformationEmedastine is a potent, high affinityhistamine H1-receptor-selectiveantagonist with Ki of 1.3 ±0.1 nM for H1-receptors while considerably weaker at H2- (K1 = 49,067 ± 11,113 nM) and H3-receptors (Ki = 12,430 ± 1,282 nM).TargetsH1 receptor

emlenoflast.

emlenoflast.

Highly potent and selective OX2antagonist: brain penetrant.

Highly potent and selective OX2antagonist: brain penetrant.

Highly potent and selective OX2antagonist: brain penetrant.

Highly potent and selective OX2antagonist: brain penetrant.