Erlotinib

UHMK1 Protein is stored in 50mM Tris-HCl, pH 7.5, 50mM NaCl, 10mM glutathione, 0.

UHMK1 Protein is stored in 50mM Tris-HCl, pH 7.5, 50mM NaCl, 10mM glutathione, 0.

InformationVarlitinib (ARRY334543) is a selective and potentErbB1(EGFR)andErbB2(HER2)inhibitor withIC50of 7 nM and 2 nM, respectively. Phase 2.In vitroARRY334543 behaves as a reversible ATP-competitive inhibitor with nanomolar potency (Ki=1 nM) both

VX-11e is a potent, selective, and orally bioavailable ERK2 inhibitor with Ki of &lt:2 nM, over 200-fold selective over other kinases tested.

inhibitor of ROCK, ERK, GSK, and AGC protein kinases.

Biochem/physiol Actions XMD17-109 is a cell-permeable, non-cytotoxic ATP site-targeting pyrimido-diazepinone derivative that acts as potent inhibitor against ERK5 (MAPK7, BMK1) kinase activity in cell-free assay (IC 50 = 162 nM: [ATP] = 50

Potent and selective ERK5 inhibitor.

InformationXMD8-85 (ERK5-IN-1) is a potent dual inhibitor of ERK5 and LRRK2 with IC50 of 87 nM and 26 nM, respectively.

InformationXMD8-85 (ERK5-IN-1) is a potent dual inhibitor of ERK5 and LRRK2 with IC50 of 87 nM and 26 nM, respectively.

InformationXMD8-85 (ERK5-IN-1) is a potent dual inhibitor of ERK5 and LRRK2 with IC50 of 87 nM and 26 nM, respectively.

InformationXMD8-85 (ERK5-IN-1) is a potent dual inhibitor of ERK5 and LRRK2 with IC50 of 87 nM and 26 nM, respectively.