Cholinergic drugs and cholinesterase inhibitors

E1R is a positive allosteric modulator of sigma-1 receptors ( Sig1R PAM ) with cognition-enhancing activity.In VitroThe only target for E1R (inhibition or enhancement of radioligand binding exceeding 20%) is the sigma receptor. 10 μM E1R does not

E1R is a positive allosteric modulator of sigma-1 receptors ( Sig1R PAM ) with cognition-enhancing activity.In VitroThe only target for E1R (inhibition or enhancement of radioligand binding exceeding 20%) is the sigma receptor. 10 μM E1R does not

E1R is a positive allosteric modulator of sigma-1 receptors ( Sig1R PAM ) with cognition-enhancing activity.In VitroThe only target for E1R (inhibition or enhancement of radioligand binding exceeding 20%) is the sigma receptor. 10 μM E1R does not

Fustinis ((±)-Fustin: 3,7,3',4'-Tetrahydroxyflavanone) is a potent amyloid β (Aβ) inhibitor. Fustinis ((±)-Fustin: 3,7,3',4'-Tetrahydroxyflavanone) increases the expression of acetylcholine (ACh) levels, choline acetyltransferase (ChAT) activity,

A competitive and reversible inhibitor of acetylcholinesterase. Antimyasthenic agent.

A peptide that selectively inhibits the activation of G q by M 1 -muscarinic cholinergic receptors. Also inhibits activation by cholecystokinin receptor in pancreatic acini at 10 &#181M.

Species : Human Assay Principle : Target Name : anti-muscarinic cholinergic receptor 3 Sensitivity : Detection Range :

A bioactive monohydroxylated metabolite of the cholinesterase inhibitor, tacrine that has less acute liver toxicity than tacrine in both animal and clinical studies of Alzheimer&rsquos disease.

A bioactive monohydroxylated metabolite of the cholinesterase inhibitor, tacrine that has less acute liver toxicity than tacrine in both animal and clinical studies of Alzheimer&rsquos disease.

A bioactive monohydroxylated metabolite of the cholinesterase inhibitor, tacrine that has less acute liver toxicity than tacrine in both animal and clinical studies of Alzheimer&rsquos disease.

A cholinesterase inhibitor that exhibits a biochemical profile very similar to tacrine.

A cholinesterase inhibitor that exhibits a biochemical profile very similar to tacrine.