Phenprobamate

A mechanism-based inactivator of human CYP2B6 (Ki = 5.6 &microM IC₅₀ = 5.1 &microM) with potent selectivity for CYP2B6 over other CYP450 isoforms.

A mechanism-based inactivator of human CYP2B6 (Ki = 5.6 &microM IC₅₀ = 5.1 &microM) with potent selectivity for CYP2B6 over other CYP450 isoforms.

Biochem/physiol Actions CP-91149 is a selective glycogen phosphorylase inhibitor. Other Notes This compound was developed by Pfizer for Kinase Phosphatase Biology research .

Biochem/physiol Actions CP-91149 is a selective glycogen phosphorylase inhibitor. Other Notes This compound was developed by Pfizer for Kinase Phosphatase Biology research .

Biochem/physiol Actions CPCCOEt is a selective non-competitive metabotropic glutamate receptor mGluR1 antagonist with no agonist or antagonist activity at mGlu2, 4a, 5a, 7b, 8a or ionotropic receptors at concentrations of up to 100 &#956:M.

Biochem/physiol Actions CPCCOEt is a selective non-competitive metabotropic glutamate receptor mGluR1 antagonist with no agonist or antagonist activity at mGlu2, 4a, 5a, 7b, 8a or ionotropic receptors at concentrations of up to 100 &#956:M.

IK1 inhibitor PA-6 (PA-6), a pentamidine analogue, is a selective and potent I K1 (K IR 2.x ion-channel-carried inward rectifier current) inhibitor, with IC 50 values of 12-15 nM for human and mouse K IR 2.x currents. IK1 inhibitor PA-6 (PA-6)

Biochem/physiol Actions JNJ-47965567 is a potent P2X7 antagonist with high affinity for the rat receptor (pKi = 8.7).

Biochem/physiol Actions JNJ-47965567 is a potent P2X7 antagonist with high affinity for the rat receptor (pKi = 8.7).

KYSE-70

InformationLoureirin B Loureirin B (LB, LrB), a flavonoid extracted from Dracaena cochinchinensis, is an inhibitor of PAI-1 with IC50 of 26.10 μM. Loureirin B downregulates p-ERK and p-JNK in TGF-β1-stimulated fibroblasts. Loureirin B promotes

InformationLoureirin B Loureirin B (LB, LrB), a flavonoid extracted from Dracaena cochinchinensis, is an inhibitor of PAI-1 with IC50 of 26.10 μM. Loureirin B downregulates p-ERK and p-JNK in TGF-β1-stimulated fibroblasts. Loureirin B promotes