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19050-50
2,3-dinor Thromboxane B2-50 ÃÆâ¦g
Price: $592.83List Price: $658.70An endogenous CB neurotransmitter that binds to both CB1 and CB2 receptors. -
62165-1
2-Arachidonyl Glycerol ether-1 mg
Price: $121.87List Price: $135.41A selective CB1 receptor agonist exhibiting Ki values of 21.2 nM and >3 µM at the CB1 and CB2 receptors, respectively more chemically stable than 2-AG, with an endogenous half-life of hours rather than minutes but 10-fold less potent than -
62165-10
2-Arachidonyl Glycerol ether-10 mg
Price: $655.07List Price: $727.86A selective CB1 receptor agonist exhibiting Ki values of 21.2 nM and >3 µM at the CB1 and CB2 receptors, respectively more chemically stable than 2-AG, with an endogenous half-life of hours rather than minutes but 10-fold less potent than -
62165-25
2-Arachidonyl Glycerol ether-25 mg
Price: $1,326.31List Price: $1,473.68A selective CB1 receptor agonist exhibiting Ki values of 21.2 nM and >3 µM at the CB1 and CB2 receptors, respectively more chemically stable than 2-AG, with an endogenous half-life of hours rather than minutes but 10-fold less potent than -
62165-5
2-Arachidonyl Glycerol ether-5 mg
Price: $371.44List Price: $412.71A selective CB1 receptor agonist exhibiting Ki values of 21.2 nM and >3 µM at the CB1 and CB2 receptors, respectively more chemically stable than 2-AG, with an endogenous half-life of hours rather than minutes but 10-fold less potent than -
11093-1
4-Quinolone-3-Carboxamide CB2 Ligand-1 mg
Price: $118.58List Price: $131.75A selective, high affinity ligand of the CB2 receptor (Ki = 0.6 nM v. CB1 binding at a Ki >10,000 nM in vitro) that may behave as an inverse agonist displays antinociceptive activity in a formalin test in mice at a dose of 6 mg/kg. -
11093-10
4-Quinolone-3-Carboxamide CB2 Ligand-10 mg
Price: $634.24List Price: $704.71A selective, high affinity ligand of the CB2 receptor (Ki = 0.6 nM v. CB1 binding at a Ki >10,000 nM in vitro) that may behave as an inverse agonist displays antinociceptive activity in a formalin test in mice at a dose of 6 mg/kg. -
11093-25
4-Quinolone-3-Carboxamide CB2 Ligand-25 mg
Price: $1,377.24List Price: $1,530.26A selective, high affinity ligand of the CB2 receptor (Ki = 0.6 nM v. CB1 binding at a Ki >10,000 nM in vitro) that may behave as an inverse agonist displays antinociceptive activity in a formalin test in mice at a dose of 6 mg/kg. -
11093-5
4-Quinolone-3-Carboxamide CB2 Ligand-5 mg
Price: $381.27List Price: $423.63A selective, high affinity ligand of the CB2 receptor (Ki = 0.6 nM v. CB1 binding at a Ki >10,000 nM in vitro) that may behave as an inverse agonist displays antinociceptive activity in a formalin test in mice at a dose of 6 mg/kg. -
11094-1
4-Quinolone-3-Carboxamide Furan CB2 Agonist-1 mg
Price: $144.91List Price: $161.01A high affinity ligand of CB2 (Ki = 8.5 nM) with little affinity for CB1 (Ki >10000 nM) demonstrates antinociceptive efficacy in the mouse formalin test at 1 mg/kg, an action which is blocked by a CB2-selective antagonist, AM630. -
11094-10
4-Quinolone-3-Carboxamide Furan CB2 Agonist-10 mg
Price: $789.30List Price: $877.00A high affinity ligand of CB2 (Ki = 8.5 nM) with little affinity for CB1 (Ki >10000 nM) demonstrates antinociceptive efficacy in the mouse formalin test at 1 mg/kg, an action which is blocked by a CB2-selective antagonist, AM630. -
11094-25
4-Quinolone-3-Carboxamide Furan CB2 Agonist-25 mg
Price: $1,724.43List Price: $1,916.03A high affinity ligand of CB2 (Ki = 8.5 nM) with little affinity for CB1 (Ki >10000 nM) demonstrates antinociceptive efficacy in the mouse formalin test at 1 mg/kg, an action which is blocked by a CB2-selective antagonist, AM630.