Controlled substance analgesic amides and amines

Application Traditionally challenging to access, this hindered amine provides a chemically differentiated building block for organic synthesis and medicinal chemistry, specifically for preparation of drug candidates containing hindered amine

3-Azidopropionic Acid contains an azide moiety and carboxylic acid group. The azide group can undergo copper-catalyzed Click Chemistry reactions with alkyne groups. The terminal carboxylic acid group can react with primary amine groups in the

3-Azidopropionic Acid contains an azide moiety and carboxylic acid group. The azide group can undergo copper-catalyzed Click Chemistry reactions with alkyne groups. The terminal carboxylic acid group can react with primary amine groups in the

3-iodo-1H-indazol-5-amine.

3-m-Tolyl-1h-pyrazol-5-amine

DescriptionTraditionally challenging to access, this hindered amine provides a chemically differentiated building block for organic synthesis and medicinal chemistry, specifically for preparation of drug candidates containing hindered amine motifs.

Application Traditionally challenging to access, this hindered amine provides a chemically differentiated building block for organic synthesis and medicinal chemistry, specifically for preparation of drug candidates containing hindered amine

DescriptionTraditionally challenging to access, this hindered amine provides a chemically differentiated building block for organic synthesis and medicinal chemistry, specifically for preparation of drug candidates containing hindered amine motifs.

4 4-DIMETHYL-2 6-DIOXO-CYCLOHEXANECARBOXYLIC ACID AMIDE-

DescriptionTraditionally challenging to access, this hindered amine provides a chemically differentiated building block for organic synthesis and medicinal chemistry, specifically for preparation of drug candidates containing hindered amine motifs.

4-[(1-oxo-7-phenylheptyl)amino]-(4R)-octanoic acid a simple amide based on (R)-α-norleucine, is a selective and potent inhibitor of sPLA2. It exhibits 95% inhibition (XI(50) = 0.003) of sPLA2 at 0.091 mole fraction without affecting the activities

Application Reactant involved in: Hydroamination-double hydroarylation for synthesis of fuzed carbazoles Cycloisomerizations of aromatic homo- and bis-homopropargylic amine / amide intermediates Asymmetric organocatalytic condensation and