Conivaptan hydrochloride

VU0364770 hydrochloride is a selective and potent positive allosteric modulator ( PAM ) of mGlu4 . VU0346770 hydrochloride exhibits EC 50 s of 290 nM and 1.1 μM at rat mGlu4 and human mGlu4 receptor , respectively. VU0364770 hydrochloride exhibits

A less active, chlorine-deficient analog of W-7, the potent calmodulin antagonist (Ki = 11 &muM) suitable for use as a control compound for understanding the specificity of other calmodulin antagonists.

A less active, chlorine-deficient analog of W-7, the potent calmodulin antagonist (Ki = 11 &muM) suitable for use as a control compound for understanding the specificity of other calmodulin antagonists.

Biochem/physiol Actions The 5-HT2C receptors have been implicated in conditions including obesity, anxiety, depression, OCD, schizophrenia, migraine, nociception and erectile dysfunction. Features and Benefits This compound was developed by

A selective 5-HT 1A receptor antagonist (pKi = 7.9-9.