-
17377-50
GSK2126458-50 mg
Price: $2,633.80List Price: $2,926.44GSK2126458 is a potent inhibitor of phosphoinositide 3-kinase isoforms (K<sub>i</sub>s = 19, 130, 24, and 60 pM for p110&alpha, &beta, &delta, and &gamma, respectively). It also inhibits mTOR in both mTORC1 and mTORC2 (K<sub>i</sub>s = 180 and -
G408838-1ml
GSK3787 (C007B-173177)
Price: $213.41List Price: $237.12InformationGSK3787 GSK3787 is as a selective and irreversible antagonist of PPARδ with pIC50 of 6.6, with no measurable affinity for hPPARα or hPPARγ.In vitroGSK3787 irreversibly antagonizes human and mouse PPARδ that covalently modifies Cys249 -
15219-10
GSK3787-10 mg
Price: $211.92List Price: $235.46A selective, irreversible antagonist of PPAR&beta/&delta (pIC<sub>50</sub> = 6.6) that inhibits the expression of PPAR&beta/&delta-regulated target genes, PDK4, CPT1a, and Angptl4. -
15219-25
GSK3787-25 mg
Price: $393.58List Price: $437.31A selective, irreversible antagonist of PPAR&beta/&delta (pIC<sub>50</sub> = 6.6) that inhibits the expression of PPAR&beta/&delta-regulated target genes, PDK4, CPT1a, and Angptl4. -
15219-5
GSK3787-5 mg
Price: $154.84List Price: $172.05A selective, irreversible antagonist of PPAR&beta/&delta (pIC<sub>50</sub> = 6.6) that inhibits the expression of PPAR&beta/&delta-regulated target genes, PDK4, CPT1a, and Angptl4. -
15219-50
GSK3787-50 mg
Price: $578.66List Price: $642.96A selective, irreversible antagonist of PPAR&beta/&delta (pIC<sub>50</sub> = 6.6) that inhibits the expression of PPAR&beta/&delta-regulated target genes, PDK4, CPT1a, and Angptl4. -
SML2024-5MG
GSK4028 (C005B-311313)
Price: $316.17List Price: $351.30Biochem/physiol Actions GSK4028 is an enantiomeric negative control for PCAF/GCN5 bromodomain inhibitor GSK4027. -
SML2024-25MG
GSK4028 (C005B-311314)
Price: $1,184.41List Price: $1,316.01Biochem/physiol Actions GSK4028 is an enantiomeric negative control for PCAF/GCN5 bromodomain inhibitor GSK4027. -
17233-10
GSK4716-10 mg
Price: $185.14List Price: $205.71A selective ERR&beta/&gamma agonist (IC<sub>50</sub> = 2 µM) that can activate the receptor with similar potency as the protein ligand, PGC-1&alpha. -
17233-50
GSK4716-50 mg
Price: $638.84List Price: $709.82A selective ERR&beta/&gamma agonist (IC<sub>50</sub> = 2 µM) that can activate the receptor with similar potency as the protein ligand, PGC-1&alpha. -
19098-25
GSK837149A-25 mg
Price: $1,233.74List Price: $1,370.82A selective, reversible inhibitor of FAS (pIC<sub>50</sub> = 7.8). -
19098-5
GSK837149A-5 mg
Price: $341.92List Price: $379.91A selective, reversible inhibitor of FAS (pIC<sub>50</sub> = 7.8).