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B413858-5mg
Brilanestrant (GDC-0810) (C09-0785-826)
Price: $216.46List Price: $240.51InformationBrilanestrant (GDC-0810, ARN-810) is a potentER-αbinder (ER-α, IC50 = 6.1 nM: ER-β, IC50 = 8.8 nM), a full transcriptional antagonist with no agonism and displays good potency and efficacy in ER-α degradation (EC50 = 0.7 nM) and MCF-7 -
B421391-1ml
Brilanestrant (GDC-0810) (C09-0786-209)
Price: $312.66List Price: $347.40InformationBrilanestrant (GDC-0810, ARN-810) is a potentER-αbinder (ER-α, IC50 = 6.1 nM: ER-β, IC50 = 8.8 nM), a full transcriptional antagonist with no agonism and displays good potency and efficacy in ER-α degradation (EC50 = 0.7 nM) and MCF-7 -
B408254-1ml
BRL-15572 Dihydrochloride
Price: $231.71List Price: $257.46InformationBRL-15572 is a5-HT1Dreceptor antagonist withpKiof 7.9, also shows a considerable affinity at 5-HT1A and 5-HT2B receptors, exhibiting 60-fold selectivity over 5-HT1B receptor.In vitroBRL-15572 displays high affinity and selectivity for -
B647605-10mg
BW 755C (C09-1113-069)
Price: $337.22List Price: $374.69BW 755C is a 5-lipoxygenase ( 5-LO ) inhibitor with an IC 50 of 5 μM. BW 755C also inhibits cyclooxygenase ( COX ) with IC 50 s of 0.65 and 1.2 μg/mL against COX-1 and COX-2 , respectivelyIn VivoBW 755C (0.03-10 mg/rat: s.c.: once) inhibits the -
B647605-5mg
BW 755C (C09-1113-070)
Price: $245.44List Price: $272.71BW 755C is a 5-lipoxygenase ( 5-LO ) inhibitor with an IC 50 of 5 μM. BW 755C also inhibits cyclooxygenase ( COX ) with IC 50 s of 0.65 and 1.2 μg/mL against COX-1 and COX-2 , respectivelyIn VivoBW 755C (0.03-10 mg/rat: s.c.: once) inhibits the -
C287028-10mg
C3 (C09-0815-503)
Price: $289.68List Price: $321.86Selective microsomal prostaglandin E synthase 1 (mPGES-1) inhibitor. -
C287028-50mg
C3 (C09-0815-504)
Price: $966.77List Price: $1,074.19Selective microsomal prostaglandin E synthase 1 (mPGES-1) inhibitor. -
14589-100
Cantharidin-100 mg
Price: $327.17List Price: $363.53Inhibits PP1 (IC<sub>50</sub> = 1.7 &muM) and PP2A (IC<sub>50</sub> = 0. -
C287880-100mg
CATPB (C09-0815-674)
Price: $6,237.94List Price: $6,931.04Product descriptionCATPB is a potent, selective free fatty acid receptor 2 (FFA2R/GPR43) antagonist. -
C287880-10mg
CATPB (C09-0815-675)
Price: $890.15List Price: $989.05Product descriptionCATPB is a potent, selective free fatty acid receptor 2 (FFA2R/GPR43) antagonist. -
C287880-25mg
CATPB (C09-0815-676)
Price: $1,926.12List Price: $2,140.13Product descriptionCATPB is a potent, selective free fatty acid receptor 2 (FFA2R/GPR43) antagonist. -
C287880-50mg
CATPB (C09-0815-677)
Price: $3,465.47List Price: $3,850.52Product descriptionCATPB is a potent, selective free fatty acid receptor 2 (FFA2R/GPR43) antagonist.