-
Add to Cart The item has been added18181-50IOX4-50 mg
Price: $1,330.94List Price: $1,478.82A selective, potent inhibitor of PHD2 (IC<sub>50</sub> = 1.6 nM) active in vivo, inhibiting prolyl hydroxylation and increasing HIF1&alpha levels in cells (IC<sub>50</sub> values range from 5. -
Add to Cart The item has been added15223-500IPBT-5CA-500 mg
Price: $376.35List Price: $418.17A selective agonist of GPR109B (HCA3 EC<sub>50</sub> = 400 nM) that displays no activity at GPR109A (HCA2). -
Add to Cart The item has been addedI649918-100mgIPN60090 dihydrochloride (C09-1140-211)
Price: $5,845.21List Price: $6,494.68IPN-60090 dihydrochloride is an orally active and highly selective inhibitor of glutaminase 1 ( GLS1 : IC 50 =31 nM), with no activity observed against GLS-2. IPN-60090 dihydrochloride exhibits excellent physicochemical and pharmacokinetic -
Add to Cart The item has been addedI649918-10mgIPN60090 dihydrochloride (C09-1140-212)
Price: $1,192.99List Price: $1,325.54IPN-60090 dihydrochloride is an orally active and highly selective inhibitor of glutaminase 1 ( GLS1 : IC 50 =31 nM), with no activity observed against GLS-2. IPN-60090 dihydrochloride exhibits excellent physicochemical and pharmacokinetic -
Add to Cart The item has been addedI649918-25mgIPN60090 dihydrochloride (C09-1140-213)
Price: $2,221.83List Price: $2,468.70IPN-60090 dihydrochloride is an orally active and highly selective inhibitor of glutaminase 1 ( GLS1 : IC 50 =31 nM), with no activity observed against GLS-2. IPN-60090 dihydrochloride exhibits excellent physicochemical and pharmacokinetic -
Add to Cart The item has been addedI649918-50mgIPN60090 dihydrochloride (C09-1140-214)
Price: $3,741.31List Price: $4,157.01IPN-60090 dihydrochloride is an orally active and highly selective inhibitor of glutaminase 1 ( GLS1 : IC 50 =31 nM), with no activity observed against GLS-2. IPN-60090 dihydrochloride exhibits excellent physicochemical and pharmacokinetic -
Add to Cart The item has been addedI649918-5mgIPN60090 dihydrochloride (C09-1140-215)
Price: $706.50List Price: $785.00IPN-60090 dihydrochloride is an orally active and highly selective inhibitor of glutaminase 1 ( GLS1 : IC 50 =31 nM), with no activity observed against GLS-2. IPN-60090 dihydrochloride exhibits excellent physicochemical and pharmacokinetic -
Add to Cart The item has been addedI339968-10mgIsosilybin B (C09-1508-945)
Price: $784.34List Price: $871.49Isosilybin B is a flavonolignan extracted from silymarin that exhibits anti-prostate cancer (PCA) activity, inhibits cancer cell proliferation, and contributes to G1-phase blockade and apoptosis.Isosilybin B induces degradation of the androgen -
Add to Cart The item has been addedI339968-1mgIsosilybin B (C09-1508-946)
Price: $274.42List Price: $304.92Isosilybin B is a flavonolignan extracted from silymarin that exhibits anti-prostate cancer (PCA) activity, inhibits cancer cell proliferation, and contributes to G1-phase blockade and apoptosis.Isosilybin B induces degradation of the androgen -
Add to Cart The item has been addedSML2098-5MGKINK-1 HYDROCHLORIDE (C15-1723-005)
Price: $421.56List Price: $468.40Biochem/physiol Actions KINK-1 (Kinase Inhibitor of NF-Κ:B-1: Bay 65-1942: CmpdA: Compound A) is an ATP-competitive, IKKβ:-selective IΚ:B kinase (IKK) inhibitor (Ki against ATP = 2 nM/IKKβ: and 135 nM/IKKα:) that potently -
Add to Cart The item has been addedSML2098-25MGKINK-1 HYDROCHLORIDE (C15-1723-006)
Price: $1,264.86List Price: $1,405.41Biochem/physiol Actions KINK-1 (Kinase Inhibitor of NF-Κ:B-1: Bay 65-1942: CmpdA: Compound A) is an ATP-competitive, IKKβ:-selective IΚ:B kinase (IKK) inhibitor (Ki against ATP = 2 nM/IKKβ: and 135 nM/IKKα:) that potently -
Add to Cart The item has been added9000249-50L-165,041-50 mg
Price: $1,226.78List Price: $1,363.09A potent and selective agonist of the nuclear receptor PPAR&beta/&delta (Ki = 9 nM, EC<sub>50</sub> ~500 nM for hPPAR&beta/&delta) less effective against PPAR&alpha and PPAR&gamma, with activity at those receptors depending on cell type and
