Rivoglitazone hydrochloride

A selective GABA_B receptor antagonist.

A selective GABA_B receptor antagonist.

General description A cell-permeable 3-aminoindazolylurea compound that acts as a potent and ATP-competitive inhibitor of VEGFR2/KDR (IC 50 = 3 nM) as well as Flt3 and cKit (IC 50 = 4 to 20 nM). Shown to block VEGF-induced VEGFR2 phosphorylation

CLP-3094 is a potent BF3 (binding function 3)-directed inhibitor of the androgen receptor (AR). CLP-3094 inhibits AR transcriptional activity (IC 50 =4 μM). CLP-3094 is a selective, potent GPR142 antagonist .In VitroCLP-3094 inhibits both an

CLP-3094 is a potent BF3 (binding function 3)-directed inhibitor of the androgen receptor (AR). CLP-3094 inhibits AR transcriptional activity (IC 50 =4 μM). CLP-3094 is a selective, potent GPR142 antagonist .In VitroCLP-3094 inhibits both an

CLP-3094 is a potent BF3 (binding function 3)-directed inhibitor of the androgen receptor (AR). CLP-3094 inhibits AR transcriptional activity (IC 50 =4 μM). CLP-3094 is a selective, potent GPR142 antagonist .In VitroCLP-3094 inhibits both an

DDR Inhibitor is a potent discoidin domain receptor (DDR) inhibitor, with an IC 50 of 3.3 nM for DDR2 , and shows 53% inhibition on DDR1 at 1.5 nM.In VitroDDR Inhibitor (Example 6) is a potent DDR inhibitor, with an IC 50 of 3.3 nM for DDR2, and

MT2receptor antagonist.

MT2receptor antagonist.

InformationdiABZI STING agonist (Compound 3) diABZI STING agonist (diABZI STING agonist-1, Compound 3) is a potent non-nucleotide STING agonist and has tremendous potential to improve treatment of cancer in humans.TargetsSTINGIn vitroIn human PBMCs,

InformationdiABZI STING agonist (Compound 3) diABZI STING agonist (diABZI STING agonist-1, Compound 3) is a potent non-nucleotide STING agonist and has tremendous potential to improve treatment of cancer in humans.TargetsSTINGIn vitroIn human PBMCs,

ApplicationOrganohalide based perovskites have emerged as an important class of material for solar cell applications. The variations/substitution in organohalide cations and anions is employed for the optimization of the band gap, carrier diffusion