-
10008647-1
11a-hydroxy Testosterone-1 mg
Price: $158.10List Price: $175.67A metabolite of testosterone, produced by CYP3A or by a mutant of CYP107A1. -
10008647-5
11a-hydroxy Testosterone-5 mg
Price: $457.56List Price: $508.40A metabolite of testosterone, produced by CYP3A or by a mutant of CYP107A1. -
13120-50
2,3-dinor Prostaglandin E1-50 ÃÆâ¦g
Price: $310.62List Price: $345.14PGE1 is not a major naturally occurring prostaglandin, but it is widely administered clinically for several indications including peripheral occlusive vascular disease, erectile dysfunction, and in neonatal cardiology. The metabolism of PGE1 is -
10009598-1
6,7-dihydroxy Bergamottin-1 mg
Price: $76.14List Price: $84.596,7-dihydroxy Bergamottin (6,7-DHB) is a potent inhibitor of CYP3A4 (IC50 = 25 µM). It appears to be the primary compound in grapefruit juice that is responsible for inhibition of testosterone 6&beta-hydrolase activity. -
10009598-10
6,7-dihydroxy Bergamottin-10 mg
Price: $359.15List Price: $399.056,7-dihydroxy Bergamottin (6,7-DHB) is a potent inhibitor of CYP3A4 (IC50 = 25 µM). It appears to be the primary compound in grapefruit juice that is responsible for inhibition of testosterone 6&beta-hydrolase activity. -
10009598-25
6,7-dihydroxy Bergamottin-25 mg
Price: $743.00List Price: $825.566,7-dihydroxy Bergamottin (6,7-DHB) is a potent inhibitor of CYP3A4 (IC50 = 25 µM). It appears to be the primary compound in grapefruit juice that is responsible for inhibition of testosterone 6&beta-hydrolase activity. -
10009598-5
6,7-dihydroxy Bergamottin-5 mg
Price: $246.75List Price: $274.176,7-dihydroxy Bergamottin (6,7-DHB) is a potent inhibitor of CYP3A4 (IC50 = 25 µM). It appears to be the primary compound in grapefruit juice that is responsible for inhibition of testosterone 6&beta-hydrolase activity. -
10008519-5
6-hydroxy Testosterone-5 mg
Price: $339.66List Price: $377.40A major metabolite produced from testosterone by the actions of CYP3A4 and CYP3A5. -
15148-10
Abiraterone Acetate-10 mg
Price: $450.18List Price: $500.20Blocks CYP17A1 by potently inhibiting both the 17&alpha-hydroxylase and the 17,20 lyase activities (IC<sub>50</sub> = 18 and 17 nM, respectively) essentially eliminates plasma testosterone while producing a 3- to 4-fold increase in plasma -
15148-25
Abiraterone Acetate-25 mg
Price: $797.91List Price: $886.57Blocks CYP17A1 by potently inhibiting both the 17&alpha-hydroxylase and the 17,20 lyase activities (IC<sub>50</sub> = 18 and 17 nM, respectively) essentially eliminates plasma testosterone while producing a 3- to 4-fold increase in plasma -
15148-5
Abiraterone Acetate-5 mg
Price: $351.26List Price: $390.29Blocks CYP17A1 by potently inhibiting both the 17&alpha-hydroxylase and the 17,20 lyase activities (IC<sub>50</sub> = 18 and 17 nM, respectively) essentially eliminates plasma testosterone while producing a 3- to 4-fold increase in plasma -
15148-50
Abiraterone Acetate-50 mg
Price: $1,532.30List Price: $1,702.55Blocks CYP17A1 by potently inhibiting both the 17&alpha-hydroxylase and the 17,20 lyase activities (IC<sub>50</sub> = 18 and 17 nM, respectively) essentially eliminates plasma testosterone while producing a 3- to 4-fold increase in plasma