Glycosidase Inhibitors

Analysis Note Assay (acidimetric): &#8805 99.0 % Melting range (lower value): &#8805 74 &#176C Melting range (upper value): &#8804 79 &#176C Identity (IR): passes test

Packaging This product may be available from bulk stock and can be packaged on demand. For information on pricing, availability and packaging, please contact Stable Isotopes Customer Service .

Packaging 1 mL in ampule This product may be available from bulk stock and can be packaged on demand. For information on pricing, availability and packaging, please contact Stable Isotopes Customer Service .

A cell-permeable aminopyrimidine compound that acts as potent, ATP-competitive, and highly selective GSK-3 inhibitor (IC 50 = 10 and 6.7 nM against GSK-3&#945 and GSK-3&#946, respectively).

A cell-permeable glycinyl hydrazone compound that acts as a potent, selective and reversible open-channel blocker of CFTR with intermediate speed (&lt1 min 95% inhibition at 50 &#181M K i = 4.3 &#181M in CFTR-expressing FRT cells for apical

A cell-permeable aminopyrimidine compound that acts as potent, ATP-competitive, and highly selective GSK-3 inhibitor (IC 50 = 10 and 6.7 nM against GSK-3&#945 and GSK-3&#946, respectively).

A cell-permeable cinnamoyl compound that reversibly inhibits P-gp (P-glycoprotein) efflux function and reverses the MDR (multidrug resistance) phenotype with no noticeable effect on P-gp expression. Shown to significantly enhance Paclitaxel- (Cat.

A cell-permeable cross-conjugated &#945,&#946-unsaturated dienone compound that induces caspase activation and apoptosis (IC 50 = 1.76 and 1.