A second-generation analog of (R)-roscovitine that inhibits Cdk1, 2, 5, and 9 (IC50s = 0.09, 0.072-0.041, 0.11, and 0.18 μM, respectively) with improved potency over its parent compound; also inhibits CK1δ/ε (IC50 = 0.40 μM) and GSK-3α/β (IC50 = 12 μM).
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- UPC:
- 51111737
- Condition:
- New
- Availability:
- 3 Days
- Weight:
- 1.00 Ounces
- HazmatClass:
- No
- WeightUOM:
- LB
- MPN:
- 14006-1
- CAS:
- 294646-77-8
- Model Number:
- C830J58
- Temperature Control Device:
- Yes