A selective, small molecule inhibitor of PIP5K1C (IC50 = 41 nM, Kd = 51 nM); decreases PIP2 membrane levels in cultured DRG neurons by 45%, significantly reducing calcium signaling; displays antinociceptive effects in mouse models of chronic pain.
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- UPC:
- 51372104
- Condition:
- New
- Availability:
- 3 Days
- Weight:
- 1.00 Ounces
- HazmatClass:
- No
- WeightUOM:
- LB
- MPN:
- 16401-5
- Model Number:
- C817Q22
- Temperature Control Device:
- Yes