AH3960 (C008B-269704)

AH3960 is a selective parathyroid hormone 1 receptor (PTHR1) agonist and also an antagonist of wild-type/T877A mutant androgen receptor (AR). AH3960 exhibits pIC50 value against wild-type PTHR1 of 4.03, the IC50 against wild-type AR of 1.5 μM, and the IC50 against T877A mutant AR of 0.35 μM. AH3960 activates the cAMP and calcium signaling pathways. AH3960 inhibits adipocyte differentiation and the expression of adipocyte markers, and promotes early differentiation of osteoblasts. AH3960 is applicable to research related to osteoporosis and prostate cancer.

Specifications & Purity: AH3960 is a selective parathyroid hormone 1 receptor (PTHR1) agonist and also an antagonist of wild-type/T877A mutant androgen receptor (AR). AH3960 exhibits pIC50 value against wild-type PTHR1 of 4.03, the IC50 against wild-type AR of 1.5 μM, and the IC50 against T877A mutant AR of 0.35 μM. AH3960 activates the cAMP and calcium signaling pathways. AH3960 inhibits adipocyte differentiation and the expression of adipocyte markers, and promotes early differentiation of osteoblasts. AH3960 is applicable to research related to osteoporosis and prostate cancer.

Grade: Moligand™

Molecular Formula: C13H22N4O3

Molecular Weight: 282.34

PubChem CID: 135508376

Isomeric SMILES: CCCCN1C(=C(C(=O)N(C1=O)CCCC)C(=N)N)O

Storage Temperature: Store at -20°C

Shipped in: Ice chest + Ice pads

UPC:

51373407

Weight:

1.09 Ounces

HazmatClass:

Yes

Quantity:

1

Unit of Measurement:

EA

WeightUOM:

LB

MPN:

A650765-1mg

Country of Origin:

China

CAS:

862907-48-0

Product Size:

1mg

Harmonized Tariff Code:

2931.90.90