CCK-B Receptor Antagonist 2 (C007B-343122)

CCK-B Receptor Antagonist 2, compound 15b, is a potent and orally active Gastrin/CCK-B antagonist with an IC 50 value of 0.43 nM. CCK-B Receptor Antagonist 2 also inhibits gastrin/CCK-A activity with an IC 50 of 1.82 μMIn VivoCCK-B Receptor Antagonist 2 (0.1 μmol/kg; intravenous injection) has an inhibition effect on pentagastrin-induced gastric acid secretion in anethsetized rats with an ED 50 of 8.3 nmol/kg . MCE has not independently confirmed the accuracy of these methods. They are for reference only.Form:SolidIC50& Target:IC50: 0.43 nM (Gastrin/CCK-B),1.82 μM (Gastrin/CCK-A). Specification: 0.98 Molecular Formula: C27H28N6O3 Molecular Weight: 484.55 PubChem CID: 23844130 Isomeric SMILES: CC(C)(C)C(=O)CN1C2=CC=CC=C2C(=N[C@H](C1=O)NC(=O)NC3=CC=CC(=C3)N)C4=CC=CC=N4

UPC:

51171830

Condition:

New

Weight:

1.06 Ounces

HazmatClass:

No

Quantity:

1

Unit of Measurement:

EA

WeightUOM:

LB

MPN:

C649841-10mg

CAS:

155412-88-7

Product Size:

10mg