GSK9311

GSK9311, a less active analogue of GSK6853, can be used as a negative control. GSK9311 inhibits BRPF bromodomain with pIC 50 values of 6.0 and 4.3 for BRPF1 and BRPF2 , respectivelyIn VitroGSK6853 is a potent (300 pM), soluble, cell active (20 nM), and highly selective inhibitor of the BRPF1 bromodomain, and demonstrates properties suitable for cellular and in vivo studies. GSK6853 is a less active analogue of GSK6853 in which the 5-amide is alkylated. MCE has not independently confirmed the accuracy of these methods. They are for reference only.Form:SolidIC50& Target:BRPF1 6.0 (pIC 50 ) BRPF2 4.3 (pIC 50 )

Specifications & Purity: GSK9311, a less active analogue of GSK6853, can be used as a negative control. GSK9311 inhibits BRPF bromodomain with pIC 50 values of 6.0 and 4.3 for BRPF1 and BRPF2 , respectivelyIn VitroGSK6853 is a potent (300 pM), soluble, cell active (20 nM), and highly selective inhibitor of the BRPF1 bromodomain, and demonstrates properties suitable for cellular and in vivo studies. GSK6853 is a less active analogue of GSK6853 in which the 5-amide is alkylated. MCE has not independently confirmed the accuracy of these methods. They are for reference only.Form:SolidIC50& Target:BRPF1 6.0 (pIC 50 ) BRPF2 4.3 (pIC 50 )

Grade: Moligand™

Molecular Formula: C24H31N5O3

Molecular Weight: 437.53

PubChem CID: 121232406

Isomeric SMILES: CCN(C1=C(C=C2C(=C1)N(C(=O)N2C)C)N3CCNC[C@H]3C)C(=O)C4=CC=CC=C4OC

Storage Temperature: Store at -20°C

Shipped in: Ice chest + Ice pads

UPC:

51373438

Weight:

1.09 Ounces

HazmatClass:

Yes

Quantity:

1

Unit of Measurement:

EA

WeightUOM:

LB

MPN:

G646258-1mg

Country of Origin:

China

CAS:

1923851-49-3

Product Size:

1mg

Harmonized Tariff Code:

2931.90.90