LAS101057 (C008B-271231)

LAS101057 is a potent, selective, and orally efficacious A2B receptor antagonist.In VivoAt 3 mg/kg, LAS101057 is active in preventing Acetyl-β-methylcholine-induced AHR, and at 10 mg/kg it inhibits AHR to Acetyl-β-methylcholine to a level virtually equal to that seen with Hexadecadrol at 1 mg/kg . MCE has not independently confirmed the accuracy of these methods. They are for reference only.Form:Solid

Specifications & Purity: LAS101057 is a potent, selective, and orally efficacious A2B receptor antagonist.In VivoAt 3 mg/kg, LAS101057 is active in preventing Acetyl-β-methylcholine-induced AHR, and at 10 mg/kg it inhibits AHR to Acetyl-β-methylcholine to a level virtually equal to that seen with Hexadecadrol at 1 mg/kg . MCE has not independently confirmed the accuracy of these methods. They are for reference only.Form:Solid

Grade: Moligand™

Molecular Formula: C18H14FN5O

Molecular Weight: 335.34

PubChem CID: 16071896

Isomeric SMILES: C1CC1C(=O)NC2=CN=C(C(=N2)C3=CN=CC=C3)C4=C(C=NC=C4)F

Storage Temperature: Protected from light;Store at -20°C;Desiccated

Shipped in: Ice chest + Ice pads

UPC:

51442306

Weight:

1.09 Ounces

HazmatClass:

Yes

Quantity:

1

Unit of Measurement:

EA

WeightUOM:

LB

MPN:

L651088-25mg

Country of Origin:

China

CAS:

925676-48-8

Product Size:

25mg

Harmonized Tariff Code:

2931.90.90