LY3154207 (C008B-271554)

LY3154207 is a potent, subtype selective, and orally available human dopamine D1 receptor positive allosteric modulator (PAM) with minimal allosteric agonist activity ( EC 50 =3 nM)In VitroIn HEK293 cells transiently expressing human, dog, rhesus monkey, and mouse D1 receptors, the EC 50 s of LY3154207 are 2.3 nM, 2.0 nM, 2.5 nM, and 62.1 nM, respectively. MCE has not independently confirmed the accuracy of these methods. They are for reference only.Form:SolidIC50& Target:EC50: 3 nM (human dopamine D1 receptor)

Specifications & Purity: LY3154207 is a potent, subtype selective, and orally available human dopamine D1 receptor positive allosteric modulator (PAM) with minimal allosteric agonist activity ( EC 50 =3 nM)In VitroIn HEK293 cells transiently expressing human, dog, rhesus monkey, and mouse D1 receptors, the EC 50 s of LY3154207 are 2.3 nM, 2.0 nM, 2.5 nM, and 62.1 nM, respectively. MCE has not independently confirmed the accuracy of these methods. They are for reference only.Form:SolidIC50& Target:EC50: 3 nM (human dopamine D1 receptor)

Grade: Moligand™

Molecular Formula: C24H29Cl2NO3

Molecular Weight: 450.40

PubChem CID: 86290953

Isomeric SMILES: C[C@H]1C2=CC=CC(=C2C[C@@H](N1C(=O)CC3=C(C=CC=C3Cl)Cl)CO)CCC(C)(C)O

Storage Temperature: Store at -20°C

Shipped in: Ice chest + Ice pads

UPC:

51373410

Weight:

1.06 Ounces

HazmatClass:

Yes

Quantity:

1

Unit of Measurement:

EA

WeightUOM:

LB

MPN:

L651647-1mg

Country of Origin:

China

CAS:

1638667-79-4

Product Size:

1mg

Harmonized Tariff Code:

2931.90.90