SB 243213

SB 243213 is a selective and high-affinity 5-HT2C receptor antagonist with a pKi of 9.37 and a pKb of 9.8 for human 5-HT2C receptor. SB 243213 shows greater than a 100-fold selectivity over a wide range of neurotransmitter receptors, enzymes and ion channels. SB 243213 has improved anxiolytic profile and has the potential for schizophrenia and motor disorders.

Specifications & Purity: SB 243213 is a selective and high-affinity 5-HT2C receptor antagonist with a pKi of 9.37 and a pKb of 9.8 for human 5-HT2C receptor. SB 243213 shows greater than a 100-fold selectivity over a wide range of neurotransmitter receptors, enzymes and ion channels. SB 243213 has improved anxiolytic profile and has the potential for schizophrenia and motor disorders.

Grade: Moligand™

Molecular Formula: C22H19F3N4O2

Molecular Weight: 428.41

PubChem CID: 443391

Isomeric SMILES: CC1=CC2=C(C=C1C(F)(F)F)N(CC2)C(=O)NC3=CN=C(C=C3)OC4=C(N=CC=C4)C

Storage Temperature: Store at -20°C

Shipped in: Ice chest + Ice pads

UPC:

51373407

Weight:

1.09 Ounces

HazmatClass:

Yes

Quantity:

1

Unit of Measurement:

EA

WeightUOM:

LB

MPN:

S647204-1mg

Country of Origin:

China

CAS:

200940-22-3

Product Size:

1mg

Harmonized Tariff Code:

2931.90.90