SB 657510

SB-657510 is a selective urotensin II (UII) receptor (UT) antagonist. The Ki values are 61, 17, 30, 65 and 56 nM for human, monkey, cat, rat and mouse receptors, respectively. SB-657510 exerts anti-inflammatory effects by inhibiting UII-induced upregulation of inflammatory mediators such as adhesion molecules, cytokines, and tissue factor in human vascular endothelial cells.Application：SB 657510 may be used to study the urotensin II receptor-mediated signaling.

Selective urotensin-II (UT) receptor antagonist

Specifications & Purity: SB-657510 is a selective urotensin II (UII) receptor (UT) antagonist. The Ki values are 61, 17, 30, 65 and 56 nM for human, monkey, cat, rat and mouse receptors, respectively. SB-657510 exerts anti-inflammatory effects by inhibiting UII-induced upregulation of inflammatory mediators such as adhesion molecules, cytokines, and tissue factor in human vascular endothelial cells.Application：SB 657510 may be used to study the urotensin II receptor-mediated signaling.

Molecular Formula: C₁₉H₂₂BrClN₂O₅S

Molecular Weight: 505.81

EC Number: 663-526-5

PubChem CID: 11272107

Isomeric SMILES: CN1CC[C@H](C1)OC2=C(C=CC(=C2)NS(=O)(=O)C3=C(C=C(C(=C3)OC)OC)Br)Cl

Storage Temperature: Store at -20°C

Shipped in: Ice chest + Ice pads

More Information: https://ald-pub-files.oss-cn-shanghai.aliyuncs.com/aladdinsci/pdp/sds/1/S287184-SCI_7f5e553cede083ed5ea36a9615b850ed.pdf

UPC:

51434931

Weight:

1.06 Ounces

HazmatClass:

Yes

Quantity:

1

Unit of Measurement:

EA

WeightUOM:

LB

MPN:

S287184-1mg

Country of Origin:

China

CAS:

474960-44-6

Product Size:

1mg

Harmonized Tariff Code:

2931.90.90

Hazard Statement Codes:

H315;H319;H335

Precautionary Statement Codes:

P261;P264;P271;P280;P321;P302+P352;P304+P340;P305+P351+P338;P362+P364;P405;P403+P233;P501;P264+P265;P337+P317;P332+P317;P319