TUG-1375 (C008B-270505)

TUG-1375 is an agonist of free fatty acid receptor 2 ( FFA2/GPR43 ), with a pK i of 6.69. TUG-1375 is inactive on FFA3, FFA4, PPARα , PPARγ , PPARδ , LXRα or LXRβIn VitroTUG-1375 exhibits pEC 50 of 7.11 in the cAMP FFA2 assay, also active on murine FFA2 orthologue (pEC 50 , 6.44 ± 0.13 in the cAMP assay). Form:SolidIC50& Target:pKi: 6.69 (FFA2)

Specifications & Purity: TUG-1375 is an agonist of free fatty acid receptor 2 ( FFA2/GPR43 ), with a pK i of 6.69. TUG-1375 is inactive on FFA3, FFA4, PPARα , PPARγ , PPARδ , LXRα or LXRβIn VitroTUG-1375 exhibits pEC 50 of 7.11 in the cAMP FFA2 assay, also active on murine FFA2 orthologue (pEC 50 , 6.44 ± 0.13 in the cAMP assay). Form:SolidIC50& Target:pKi: 6.69 (FFA2)

Grade: Moligand™

Molecular Formula: C22H19ClN2O4S

Molecular Weight: 442.92

PubChem CID: 138319694

Isomeric SMILES: CC1=C(C(=NO1)C)C2=CC=C(C=C2)C(=O)N3[C@@H](CS[C@@H]3C4=CC=CC=C4Cl)C(=O)O

Storage Temperature: Store at -20°C

Shipped in: Ice chest + Ice pads

UPC:

42292304

Weight:

1.09 Ounces

HazmatClass:

Yes

Quantity:

1

Unit of Measurement:

EA

WeightUOM:

LB

MPN:

T649206-1mg

Country of Origin:

China

CAS:

2247372-59-2

Product Size:

1mg

Harmonized Tariff Code:

2931.90.90